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2-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
9-ethyl-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-phenoxypropan-1-one
2-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenyl)ethan-1-amine
2-phenoxy-N-[(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
methyl 1-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)-2-hydroxypropyl]piperidine-4-carboxylate
methyl 3-{[1-(3-phenylpropyl)piperidin-3-yl]carbamoyl}propanoate
3-(5-acetylpyridin-2-yl)-4H-chromen-4-one
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-ethyl-5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-amine
3-(2-aminoethyl)-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,5S)-5-(3-fluorophenoxymethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
3-[(3R,4S)-1-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[1-(methoxymethyl)cyclopentyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-3-(2-methyl-5-oxopyrrolidin-2-yl)-N-{[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}propanamide
3-{[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]methyl}pyridine
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})(oxolan-2-ylmethyl)amine
(2S)-3-phenyl-2-(quinoxalin-6-ylformamido)propanamide
N-[3-(1,3-benzothiazol-2-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}thieno[2,3-d]pyrimidine-6-carboxamide
2-(3,4-difluorophenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3R,5S)-5-(morpholine-4-carbonyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
5-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-[4-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]pyridine
{4-methyl-5-[(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)methyl]-4H-1,2,4-triazol-3-yl}methanol
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-1H-indole-3-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}thiolan-3-amine
methyl (2R,4S)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-hydroxypiperidine-2-carboxylate
5-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-[(benzyloxy)methyl]-1-[(2S)-oxolan-2-ylmethyl]-1H-1,2,3-triazole
2-{4-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}-N,N-dimethylacetamide
(1S,5R)-3-(3-phenylpropyl)-6-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
2-(2H-1,3-benzodioxol-5-yl)-N-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]azepan-4-yl}acetamide
methyl 1-methoxy-2-oxo-8-(quinoxalin-5-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(4-ethynylphenyl)methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
1-[(2-chlorophenyl)methyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-chloro-N-(1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1,2-oxazolidin-4-ol
1-[(9-ethyl-9H-carbazol-3-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
N-(3-methoxyphenyl)-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)propanamide
2-(3-acetyl-1H-indol-1-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)acetamide
2-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]propan-1-one
1-[(2-fluorophenyl)methyl]-1-(2-hydroxyethyl)-3-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
methyl 3-{[(3aR,6aS)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]amino}-4-methoxybenzoate
5-methoxy-2-{[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol