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(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2-ethylpyrimidine-5-carboxamide
N-[(2-chlorophenyl)methyl]-3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}propanamide
6-(2,4-dimethoxyphenyl)-2,4-dimethylpyridine-3-carbonitrile
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2,5-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 1-[2-hydroxy-3-(3-{[(3-hydroxypropyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-[(2-methoxyethyl)(methyl)sulfamoyl]benzamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
propan-2-yl 1-methyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-butyl-N-[(2-methylphenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidin-2-one
6-(2,3-dihydro-1H-inden-2-yl)-3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(3-fluorophenyl)-6-(4-methyl-1,3-oxazole-5-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl 6-(2-ethylbutanoyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3-fluoro-4-methylphenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(3-methoxybenzoyl)piperazine
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]pent-4-enamide
2-{[4-(6-methoxypyridazin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
4-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-(1-benzofuran-2-ylmethyl)-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
methyl 2-{[1-(diphenylmethyl)-1H-1,2,3-triazol-4-yl]formamido}-4-(methylsulfanyl)butanoate
4-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-1-(4-methylbenzoyl)piperidine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidin-4-amine
4-[(4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-(furan-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{4-methyl-5-[(1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4H-1,2,4-triazol-3-yl}methanol
1-[2-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-chloro-N-(4-{4-[(2-methylpropyl)amino]piperidin-1-yl}phenyl)benzamide
5-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-({7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
N-cyclopropyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)phenyl]acetamide
(3R,4S)-N,N-dimethyl-1-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(propan-2-yl)pyrrolidin-3-amine
1-(1-methylpiperidin-4-yl)-4-[3-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-butoxy-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
4-(2,3-dihydro-1H-isoindol-2-yl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-1,3-oxazole-4-carboxamide
N-methyl-N-(prop-2-en-1-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
(1R,3S)-3-({[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}carbamoyl)cyclopentane-1-carboxylic acid
2-(3-methoxyphenyl)-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
{3-[(3-chlorophenyl)methyl]-1-[2-(dimethylamino)benzoyl]piperidin-3-yl}methanol
2-[({1-[(4-chlorophenyl)methyl]-1H-pyrazol-5-yl}carbamoyl)amino]-N-(propan-2-yl)acetamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-ol
N-(5-chloro-2-methylphenyl)-N'-{2-[(pyridin-3-yl)amino]ethyl}propanediamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}){[1-(propan-2-yl)pyrrolidin-3-yl]methyl}amine
1-(4-chloro-2-fluorobenzoyl)-3-(2-methoxyphenoxy)azetidine
5-(2,4-difluorophenoxymethyl)-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,2-oxazole-3-carboxamide