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N-[1-(6-methylpyridin-2-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
[(3R,4R)-1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(3S,4S)-1-(4-methoxybenzoyl)-4-[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyrrolidin-3-ol
N3,N3-diethyl-1-[2-(4-methoxyphenyl)ethyl]-N5-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
dimethyl({2-[4-(4-phenyl-1H-imidazole-5-carbonyl)morpholin-2-yl]ethyl})amine
8-[(2-chlorophenyl)methyl]-3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,4-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
3-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-2,3-dihydro-1H-inden-1-one
1-benzyl-3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
(1R,5R)-3-benzoyl-6-[(4-fluoro-3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N'-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}butanediamide
4-[2-(2-oxopyrrolidin-1-yl)propanoyl]-1-phenylpiperazin-2-one
4,6-dimethyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrimidin-2-amine
N-cyclopropyl-2-fluoro-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-sulfamoylbenzamide
3-(2-methoxyphenyl)-1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
N-({1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-hydroxyazepan-4-yl}methyl)methanesulfonamide
2-ethoxy-4-(1-{2-[(pyridin-3-yl)amino]ethyl}-1H-imidazol-2-yl)phenol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-1H-indazole-3-carboxamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzenesulfonamide
N-ethyl-N-(4-hydroxybutyl)-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)morpholine-2-carboxamide
3-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-fluoro-N-(3-oxo-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propyl)benzamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-phenoxyethan-1-one
4-chloro-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-ethyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
(4aS,7aR)-1-(4-chlorobenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-(quinoxalin-2-yl)pyrrolidin-3-amine
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl][(8-methoxy-2H-chromen-3-yl)methyl]methylamine
benzyl[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-1-[3-(1,3-oxazol-5-yl)phenyl]piperidine
3-(5-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
1-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-1-(thiophen-3-ylmethyl)piperidine
(5S,9aS,9bS)-5-[2-(prop-2-en-1-yloxy)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{4-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenyl}methanol
(1R,5S,6R)-3-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
4-{[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]sulfonyl}-N-methyl-N-(prop-2-en-1-yl)benzamide
4-benzyl-1-(4,6-dimethylpyrimidin-2-yl)-3-ethyl-1,4-diazepan-5-one
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(5-methoxy-1H-indol-2-yl)methyl]amine
1-(4-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-4-oxobutyl)pyrrolidin-2-one
4,5-dimethyl-6-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-[(2-chlorophenyl)methyl]-5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione