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N-(2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}ethyl)aniline
2-[benzyl(methyl)amino]-N-(2,3-dihydroxypropyl)-2,3-dihydro-1H-indene-2-carboxamide
2-methoxy-5-({methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amino}methyl)benzoic acid
5-methyl-4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
8-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-({1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)propanoate
7-(2,3-dimethoxyphenyl)-9-methoxy-4-(3-phenylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
3-(3-fluorophenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
1-{2-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
diphenyl[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]methanol
N-[(2-fluorophenyl)methyl]-2-(morpholin-4-yl)-6-phenylpyridine-3-carboxamide
N-[(2R,3R)-1'-[2-(2-fluorophenyl)acetyl]-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-[(4-fluorophenyl)methyl]-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
4-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-3-phenyl-1H-pyrazole-5-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-2-carboxamide
N-[3-(4-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
N-(1-hydroxybutan-2-yl)-2-methoxy-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide
1-[7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinoline-4-carbonyl]piperidine-3-carbonitrile
1-{[3-(1,2-oxazinane-2-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-indole
1-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2,3,5,6-tetramethyl-N-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}benzamide
2-[(1H-imidazol-2-ylmethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
2-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
3-(5-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)azepan-2-one
4-(5-{1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carbonyl)piperazin-2-one
2-methyl-8-[(3-phenyloxolan-3-yl)methyl]-2,8-diazaspiro[4.5]decane
5-(azocane-1-carbonyl)-2-[(phenylsulfanyl)methyl]pyrimidin-4-ol
N-{1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
N-(3-methoxypropyl)-6-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(1-{[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}cyclopropyl)methanol
2-[(1-hydroxycyclohexyl)methyl]-4-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N5-tert-butyl-1-cyclohexyl-N3-[(3-methoxyphenyl)methyl]-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(diphenylmethyl)piperazine
1-(3-chloro-4-fluorobenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
8-methyl-4-(2-methylpiperidine-1-carbonyl)-2-(2-methylpyrimidin-5-yl)quinoline
N-(2,4-dimethoxyphenyl)-3-[1-(3-methoxypropanoyl)piperidin-4-yl]propanamide
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
methyl 4-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]butanoate
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methyl-2-propylpyrimidine
ethyl 1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-[4-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]pyridine-4-carbonitrile
7-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
7-(2-hydroxyethyl)-2-[3-(2-methyl-1H-indol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-(3-methoxyphenyl)-N-[3-(morpholin-4-yl)propyl]-1,2,4-triazin-3-amine
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-(1H-indol-3-yl)acetamide
N-benzyl-N-methyl-3-{[methyl(propan-2-yl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-4-phenyl-1,3-thiazole