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ethyl 5-(2,2-dimethyloxane-4-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2,5-thiadiazole
2-[4-(3-fluorobenzenesulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
N-(1-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
ethyl 1-[2-(cyclohex-1-en-1-yl)acetyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-(methylsulfanyl)acetamide
methyl 4-[5-oxo-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]butanoate
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(4-methyl-1,3-thiazol-2-yl)benzamide
1-(2-chlorophenyl)-4-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methylpyrazin-2-yl)methyl]piperidin-2-one
8-(1,3-thiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
3-(1,3-thiazol-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aR)-6-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
5-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(3-methoxypropyl)-1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidine
3-(prop-2-en-1-yl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidine-3-carboxylic acid
8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]benzonitrile
1-[1'-(5-ethylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
7-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-{[4-(2,4-dimethylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-ethoxypropan-1-one
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(1-methyl-1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-(3-phenylpropyl)-1H-imidazol-2-yl]pyridine
(3-{5-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(thiophen-2-yl)acetamide
methyl 2-[(1-cyclohexyl-1H-1,2,3-triazol-4-yl)formamido]-4-(methylsulfanyl)butanoate
2-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyridine-4-carbonitrile
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(pyridin-4-yl)ethyl]acetamide
N-[(2,4-dichloro-6-methylphenyl)methyl]-1-(methoxymethyl)cyclopropane-1-carboxamide
3,5,7-trimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1H-indole-2-carboxamide
N-(1-{1-[2-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
(2E)-3-(furan-2-yl)-1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]prop-2-en-1-one
N-[4-(2-fluorophenoxy)phenyl]-1-(pyridine-3-carbonyl)piperidine-2-carboxamide
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-indazole
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
2-[(4-methoxyphenyl)methyl]-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]morpholine
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}butanamide
4-fluoro-3-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]benzene-1-sulfonamide
(1-{[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
2-methyl-N-[2-(oxan-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-cyclopentyl-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
3-(2-chloro-4,6-dimethylphenyl)-1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
N-[1-({[(2-methoxyphenyl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]thiophene-3-carboxamide
1-[(4-ethoxyphenyl)methyl]-3-(2-methoxybenzoyl)piperidine
N-({7-[4-(4-fluorophenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(pyrrolidin-1-yl)acetamide
N1-(piperidin-3-yl)-N2-(pyridin-3-yl)ethane-1,2-diamine
1-(3-methoxyphenyl)-3-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methylurea