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1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(morpholin-4-yl)ethan-1-one
2-(4-ethylpiperazin-1-yl)-N-[(3-methylphenyl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(3,3-diphenylpiperidine-1-carbonyl)-6-methylpyridine
3-[2-(1H-pyrazol-1-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(3-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-methoxy-5-[3-(1-methoxyethyl)phenyl]benzamide
2-(2-hydroxypropyl)-9-(1-methyl-1H-pyrazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-acetyl-3-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
N-[(3S,4R)-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1,3-benzothiazol-2-amine
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
(2-methoxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-1-methylazepane-2-carboxamide
3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
4-methyl-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
1-(4-fluorophenyl)-N-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl][(5-ethylpyridin-2-yl)methyl]methylamine
4-{3-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2,2-dimethylpropyl}morpholine
N-[2-(thiophen-2-yl)ethyl]-2-(trifluoromethyl)morpholine-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(3R,4S)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-methyl-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]thian-4-amine
N-{[(1R,2R)-2-hydroxy-2-methylcyclohexyl]methyl}-3-(3-hydroxy-3-methylbutyl)benzamide
N-[(2R,3R)-2-methoxy-1'-[4-(2-methylpropyl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
4-{4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}amine
1-methyl-N-(pyridin-3-ylmethyl)-N-(1,3-thiazol-4-ylmethyl)piperidin-4-amine
1-[2-(3-fluorophenyl)ethyl]-N-[(6-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-{[3-(2-methoxyethoxy)phenyl]methyl}-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-methoxy-1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-2-carboxamide
1-benzyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,2-dimethyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
(4-benzyl-1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}benzamide
(3S,4S)-4-(morpholin-4-yl)-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-3-ol
1-(2-methoxyphenyl)-4-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}piperazine
(1R,5R)-N,N-dimethyl-6-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-cyclopropyl-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-fluorophenyl)methyl]piperidine
(4aS,8aR)-1-propyl-6-[3-(pyridin-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
methyl 4-{[(2S,4R)-2-(dimethylcarbamoyl)-4-(pyridin-2-ylsulfanyl)pyrrolidin-1-yl]methyl}benzoate
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(3-methoxybenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
1-({6-[5-chloro-2-(propan-2-yloxy)phenyl]pyridin-3-yl}methyl)-4-methylpiperazine
(4aS,7aR)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione