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(3R,4R)-4-(hydroxymethyl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidin-3-ol
ethyl 3-benzyl-1-{[4-(methoxycarbonyl)phenyl]carbamoyl}piperidine-3-carboxylate
1-phenyl-N-{3-[(pyridin-3-yl)amino]propyl}-1H-1,2,3-triazole-4-carboxamide
5-[2-(3,4,5-trimethoxyphenyl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-cyclopentyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-5-oxopyrrolidine-3-carboxamide
[(3R,4R)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
5-chloro-2-(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-methyl-4-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-imidazole
1-[(2,6-difluoro-3-methoxyphenyl)methyl]-5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazole
2-(4-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}quinazolin-2-yl)ethan-1-amine
7-[3-(2-methylphenyl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N-ethyl-N-(pyridin-4-ylmethyl)-1-(quinoxaline-6-carbonyl)piperidin-3-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
N-(2-{4-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]phenoxy}ethyl)acetamide
1-[(2-fluorophenyl)methyl]-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-6-oxopiperidine-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]-N-methylacetamide
methyl 3-(1-benzofuran-2-carbonyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
N-cyclohexyl-N-ethyl-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
6-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-2-methylpyrimidin-4-ol
3-hexyl-8-(1-methyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-(trifluoromethyl)benzamide
[(3R,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[3-(2-methylpropyl)-1,2-oxazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
2-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(4-fluorophenyl)propan-1-one
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)pyrrolidine-2,5-dione
2-ethyl-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(2-fluorophenyl)piperidine-1-carboxamide
1-methanesulfonyl-3-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}piperidine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-4-(morpholin-4-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]cyclopropane-1-carbonitrile
9-[(2,5-dimethylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(piperidine-1-carbonyl)piperidine
3-[(1-methylpyrrolidin-3-yl)methyl]-1-(4-phenoxyphenyl)urea
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
7-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[(3-methoxyphenyl)amino]butanamide
[(2-cyclohexylpyrimidin-5-yl)methyl][(5-cyclopropyl-1H-pyrazol-3-yl)methyl]methylamine
8-(1H-imidazol-1-yl)-2-methylquinolin-4-ol
3-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
N,N-dimethyl-5-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}pyrimidin-2-amine
1-[2-(furan-2-yl)pyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1-(9H-purin-6-yl)piperidin-4-amine
4-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one