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(4aR,7aS)-1-cyclopropanecarbonyl-4-(2-methoxy-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
ethyl 4-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)piperidine-1-carboxylate
2-({2-amino-6-[6-(benzyloxy)pyridin-3-yl]pyrimidin-4-yl}amino)ethan-1-ol
(2R,3R,6R)-5-cyclopropanecarbonyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[4-(2-amino-1,3-thiazol-4-yl)phenyl]benzamide
ethyl 2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}acetate
6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)azetidin-3-yl]-2-methylpiperidine
(propan-2-yl)({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-chloro-1-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(thiophen-2-yl)ethan-1-one
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]propanamide
methyl 2-({[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate
3-[4-(3-hydroxyphenyl)piperidin-1-yl]-N-(pyridin-3-yl)propanamide
2,8-dimethyl-N-[2-(4-methylmorpholin-2-yl)ethyl]quinoline-4-carboxamide
(3S,4R)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-[1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-2-phenylethyl]-N-methylpyridine-2-carboxamide
N-[(4-methylphenyl)methyl]-5-(phenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
3-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
1-benzyl-5-{[2-(diethylamino)ethyl](methyl)amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(2-methylphenyl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
8-(2-phenoxybenzoyl)-1-oxa-8-azaspiro[4.5]decane
4-{1-[(4-methoxyphenyl)amino]cyclopentanecarbonyl}piperazine-2-carboxylic acid
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine
1-[2-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N6-(2-methoxyethyl)-N5-methyl-N5-[3-(piperidin-1-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
N-cyclopropyl-3-(5-methylfuran-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethyl-1,3-thiazol-2-amine
2-(2-chloro-4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)acetamide
3-({[1-(morpholine-4-carbonyl)piperidin-4-yl]carbamoyl}amino)benzamide
N-ethyl-N-[(2-fluorophenyl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
5-oxo-N-(pentan-3-yl)-N-(2-phenylethyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
2-{[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}benzonitrile
1-[(4,5-dimethylfuran-2-yl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
3-{4-phenyl-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}propan-1-ol
5-cyclopropyl-N-(3-methoxypropyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-methyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N5-benzyl-N6-[(2-methyl-1,3-thiazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-[1-(2,2-dimethylpropyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)-1-phenylpiperazin-2-one
(5S,9aS,9bS)-2-phenyl-5-(2,3,4-trimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{5-[4-(piperidin-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N,N-dimethyl-1-[3-(piperidin-4-ylmethyl)benzoyl]azepan-4-amine