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3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(piperidin-1-yl)propan-1-one
1-(3-{[1,2,4]triazolo[4,3-a]pyrazin-3-yl}-1H-indol-1-yl)ethan-1-one
1-ethyl-4-({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperazin-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-(2-methyl-1-benzofuran-7-yl)-1,4-diazepane-1-carboxamide
3-(1-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-1,2,3-triazol-4-yl)benzonitrile
2-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
3-(3,4-dimethoxybenzoyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
5-hydroxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrazine-2-carboxamide
3-methyl-7-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3E)-1-{2-[5-(4-methyl-1,4-diazepane-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}pent-3-en-1-one
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
6-tert-butyl-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)(methyl)(pyridin-2-ylmethyl)amine
N-(2-hydroxyethyl)-N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
3-ethyl-5-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-1,2-oxazole-4-carboxamide
methyl (2S,4S)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(3-ethoxy-2-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3aR,6aR)-2-benzyl-N-[(6-hydroxypyrimidin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]-6,7-dimethoxy-1,2-dihydroquinolin-2-one
1-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,3-benzodiazole-6-carboxylate
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-(2-methylpropyl)-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepane
N'-(2,5-dimethylphenyl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]propanediamide
2-(2,4-dichlorophenoxy)-N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-[1-(pyridin-3-yl)propan-2-yl]acetamide
2-(2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
2-[5-(1-benzyl-1H-pyrazol-4-yl)-3-cyclopentyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(piperazin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
(3S)-3-ethyl-4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholine
6-{2-[(4-methoxyphenyl)methyl]morpholine-4-carbonyl}quinoxaline
(2S,4R)-4-[2-(2,4-difluorophenyl)acetamido]-1-(furan-3-ylmethyl)-N-methylpyrrolidine-2-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[(2E)-3-phenylprop-2-enoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-butyl-5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-1,3-benzoxazole
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)oxolane-3-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
5-(dimethylamino)-2-[2-(2-ethylphenoxy)ethyl]-2,3-dihydropyridazin-3-one
7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(6-methylpyridin-3-yl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazine-2-carboxamide
N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(4-chloro-1H-pyrazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
4-chloro-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrrole-2-carboxamide
3-(3-methylbut-2-en-1-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine-3-carboxylic acid
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[1-(propan-2-yl)pyrrolidin-2-yl]methyl}propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(dimethyl-1,2-oxazol-4-yl)-N-methylpropanamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,4-dimethyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide