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1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}azepan-4-amine
2-(2,3-dimethoxyphenyl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
[5-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)-2-ethoxyphenyl]methanol
(5R)-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
3-(azepane-1-carbonyl)-N-methyl-N-(2-methylpropyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2,5-dihydro-1H-pyrrole-2-carboxamide
(1R,3S)-3-{[2-(2,3-dihydro-1H-indol-1-yl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
4-(4-{[(3-fluorophenyl)methyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-1-methylazepane-2-carboxamide
methyl 3-(2-benzylmorpholine-4-carbonyl)benzoate
3-chloro-N-cyclopentyl-4-{[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-[(3S,4R)-1-cycloheptyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
4-benzoyl-1-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperidine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methoxyfuran-2-carboxamide
5-{[4-(4-ethyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]methyl}-2-hydroxybenzoic acid
(1S,4S)-2-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
1-(3-methoxy-4-methylphenyl)-3-(2-methoxyethyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-benzyl-1-[(3,4-dimethoxyphenyl)methyl]-N-methylpiperidin-3-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-[(pyridin-4-ylmethyl)amino]pyridine-3-carboxamide
4-(2-methoxypyridine-3-carbonyl)-3,4-dihydro-2H-1,4-benzoxazine
1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-benzyl-8-(9H-purin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-amino-3-ethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
4-(4-fluorophenyl)-1-(4-methylpyrimidin-2-yl)piperidin-4-ol
1-[(diethylcarbamoyl)methyl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(2S)-2-amino-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-(4-hydroxyphenyl)propan-1-one
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(4-methylphenyl)sulfanyl]propanamide
2-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)benzoic acid
N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-methyl-8-(3-methyl-1-benzothiophene-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2,5-difluoro-N-(1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-2-(5-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
N,N,4-trimethyl-5-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-amine
7-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-[(3-chlorophenyl)methyl]-N-(pyrimidin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
(1S,5R)-3-benzyl-N-(2-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-(furan-3-carbonyl)-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
3-cyclopropyl-N-[(2-phenoxypyridin-3-yl)methyl]-1H-pyrazole-5-carboxamide
4-cyclopentyl-N-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-oxopiperazine-1-carboxamide
2-[(5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetic acid
4-({3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
N-{4-[2-(furan-2-yl)-2-oxoacetamido]phenyl}-5-methylfuran-2-carboxamide
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-1-methylpiperidine-4-carboxamide
2-methoxy-N-[(8-{[3-(2-methylphenyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide