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2-(dimethylamino)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(2R,3R)-3-amino-1'-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(3-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-2-(4-methyl-2-oxopyrrolidin-1-yl)acetamide
2-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-N-propylaniline
3-(aminomethyl)-4-(5-chloro-2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
N-(4-acetylphenyl)-3-[2-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
2-[(4aR,7aS)-4-[(5-ethylpyridin-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(4aS,8aR)-6-(1-methyl-1H-pyrazole-3-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-(methoxymethyl)-N-[4-(5-methyl-4-{[3-(4-methylphenyl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-1-methyl-2-phenylpiperazine
N-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
4-(4-chlorophenyl)-3-(ethoxymethyl)-4H-1,2,4-triazole
methyl (2S)-1-{2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]acetyl}pyrrolidine-2-carboxylate
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(5-methylfuran-2-yl)methyl]benzamide
1-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-chloro-4-hydroxy-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}quinoline-3-carboxamide
4-{5-[1-(furan-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}thiomorpholine
2-(2,5-difluorophenyl)-N-{[8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
methyl 1-(2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperidine-2-carboxylate
4-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}azetidin-3-yl)morpholine
4-(2-methyl-1H-imidazol-1-yl)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
1-(1-benzothiophen-5-ylmethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-{1-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
5-(4-cyclohexylphenyl)-N-(1,2-oxazol-3-ylmethyl)-1,2,4-triazin-3-amine
2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-4-carboxamide
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(1,3-thiazol-2-yl)piperidine
1-(naphthalen-1-ylmethyl)-4-[(propan-2-yl)amino]pyrrolidin-2-one
8-(2,2-dimethylpropyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-phenyl-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
3-[4-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-3-carboxamide
2,6-dimethyl-N-{3-[methyl(phenyl)amino]propyl}pyridine-4-carboxamide
6-methyl-3-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
5-(2-methoxyacetamido)-N-[2-(2-methoxyphenyl)ethyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(4aR,8aS)-1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
N-[1-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
N'-cyclopentyl-N'-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-N,N-dimethylbutanediamide
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(ethanesulfonyl)piperidine
N-[(1-benzylpiperidin-4-yl)methyl]-1-ethyl-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
ethyl 1-(2,4-dimethylbenzenesulfonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-chloro-6-methoxy-4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
5,6-dimethyl-2-(3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one