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2-{1-[1-(5-chloronaphthalene-1-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
2-cyclopropyl-4-hydroxy-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
3,5-dimethyl-N-{3-methyl-1-[7-(3-methylfuran-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
N-({2-[4-(furan-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
5-chloro-2-methoxy-4-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenol
3-[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]cyclopentan-1-one
2-[benzyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
8-[2-(3,4-dimethylphenoxy)ethyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)thiophene-2-carboxamide
1-methyl-4-[3-(4-methylphenyl)-3-phenylpropanoyl]piperazin-2-one
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-(1-benzylpiperidin-4-yl)-5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)imidazolidine-2,4-dione
2-amino-4-{2-[3-(dimethylamino)propoxy]phenyl}-6-(1-methylcyclopropyl)pyridine-3-carbonitrile
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]oxane-4-carboxamide
3-{[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N,1-dimethyl-6-oxo-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,6-dihydropyridazine-3-carboxamide
(2S)-2-[(5-ethanesulfonamido-1-methyl-2-phenyl-1H-1,3-benzodiazol-7-yl)formamido]-3-methylbutanamide
[(2S,4R)-4-(dimethylamino)-1-{1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}pyrrolidin-2-yl]methanol
2-({[(3R,4R)-1-(4-ethylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-{3-[({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
N-({7-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
1-[(4-methylphenyl)methyl]-4-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
2-{4-phenyl-1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-5-yl}-1H-indole
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
9-[(2R)-2-hydroxy-2-phenylethyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)cyclobutanamine
6-[(diethylamino)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S)-2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}propanamide
1-cyclopentyl-N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]piperidine-4-carboxamide
methyl (2S)-1-[2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carbonyl]pyrrolidine-2-carboxylate
3-(4-methoxyphenyl)-1-(morpholin-4-yl)-3-phenylpropan-1-one
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-(3-fluorophenyl)-6-(5-methyl-1,2-oxazole-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1,2-oxazol-3-ylmethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
{1-[2-(4-fluorophenoxy)ethyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
1-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
3-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]-N-methylethane-1-sulfonamide
4-[(2,4-dimethoxyphenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine-2-carboxamide
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carboxamide
1-[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
N-(2,4-dimethylphenyl)-2-[(2-phenoxyethyl)amino]acetamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
1-{1-[(ethylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-ethoxy-5-(2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyrimidin-4-yl)benzoic acid