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(3S,4R)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-(2-methoxyethyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carboxamide
9-(5-fluoropyrimidin-2-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-ethoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-(3-acetylphenoxymethyl)-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-2H-1,3-benzodioxole-5-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-(2-methylpropyl)-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
5-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethyl)piperazine
1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(pyridin-3-yl)propan-1-one
N-cyclopentyl-1,3-dimethyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1H-pyrazole-5-carboxamide
1-methyl-4-{1-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl}piperazine
N-[2-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenoxy)ethyl]acetamide
3-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(2-phenylethyl)piperidine-3-carboxamide
N-(2-methanesulfonylethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-{3-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]propyl}-1H-indole
{5-fluoro-7-[3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-(2-aminoethyl)-N,5,6-trimethyl-N-[4-(morpholin-4-yl)butyl]thieno[2,3-d]pyrimidin-4-amine
N-[2-(1H-indol-3-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
1-[1-(2-hydroxy-4-methylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
2-{4-[(2,5-difluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-benzyl-3-ethyl-1-[3-(1H-pyrazol-1-yl)propanoyl]-1,4-diazepan-5-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazine
N-methyl-3-[1-(pyrazin-2-yl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]acetamide
[3-(2-methoxyethyl)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-3-yl]methanol
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,6-dimethylpyrimidine-4-carboxamide
3-methyl-1-(4-{5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)-1H-pyrazol-5-amine
2-methanesulfonamido-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
{3-[(2-fluorophenyl)methyl]-1-[2-(3-methylphenyl)benzoyl]piperidin-3-yl}methanol
3-methoxy-2-[(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
N-[(3R,4R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-{4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}pyrimidine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(5,6-dimethylpyrimidin-4-yl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
5-(cyclopentylamino)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[5-(2,1,3-benzothiadiazol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
[(4-fluorophenyl)methyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
3-(4-benzylpiperazine-1-carbonyl)-2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
2-methoxy-4-{1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-imidazol-2-yl}phenol
2,6-difluoro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzene-1-sulfonamide
N-({1-[(9-ethyl-9H-carbazol-3-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide