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(1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[(3-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-2-ethyl-N-(oxolan-2-ylmethyl)butanamide
(5S,9aS,9bS)-5-(6-chloro-2H-1,3-benzodioxol-5-yl)-2-[(3-chlorophenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]propan-1-one
1-(4-ethylpiperazin-1-yl)-3-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}propan-1-one
1-(morpholine-4-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
1,9-dimethyl-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[(2S,4S)-4-fluoro-1-[2-(methylsulfanyl)acetyl]pyrrolidin-2-yl]methyl}-2-(4-methoxyphenyl)acetamide
N-[1-(1-benzothiophen-2-ylmethyl)pyrrolidin-3-yl]acetamide
3-(3-chloro-4-methoxyphenyl)-4-methylpyridine
2-(4-fluorophenyl)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidine
(3S,4R)-1-{2-[methyl(phenyl)amino]acetyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenoxyethan-1-one
N-(1-benzothiophen-5-ylmethyl)-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
7-(6-aminopyridine-3-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-fluoro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
N,N-dimethyl-4-[4-(4-propylpiperazine-1-carbonyl)phenoxy]piperidine-1-sulfonamide
(3S,9aR)-3-benzyl-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(4-{[methyl(oxan-2-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
7-acetamido-1-[(4-fluorophenyl)methyl]-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-{[2-(cyclopentyloxy)phenyl]methyl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2,6-dimethylquinoline-4-carboxamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
methyl 1-{[4-(7-fluoro-2-methylquinoline-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-2-carboxylate
(3aR,7aS)-5-methyl-2-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-1,2-dihydrophthalazin-1-one
N-(1-{7-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-(dimethylamino)acetamide
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrazine-2-carboxamide
2-(4-methoxyphenoxy)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
6-methoxy-3-methyl-N-{3-[(pyridin-3-yl)amino]propyl}-1-benzofuran-2-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(8-methylquinolin-5-yl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
6-(2,5-dimethylphenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)propan-1-ol
4-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-5-[3-(trifluoromethyl)phenyl]pyrimidine
(4aS,7aR)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-N-phenyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
2-(oxolan-2-ylmethyl)-9-[6-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2E)-1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(3-fluorophenyl)prop-2-en-1-one
1-benzyl-5-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N-diethyl-3-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}benzamide
5-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
5-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione