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3-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-2-(thiomorpholin-4-yl)acetic acid
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-cyclohexyl-3-({[(2-fluoro-5-methoxyphenyl)methyl]amino}methyl)-N-methylpyridin-2-amine
ethyl 1-[3-(1H-pyrazol-1-yl)propyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
N-benzyl-4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(2S,4S)-4-(2-ethoxyacetamido)-N,N-diethyl-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N,N-diethylacetamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-cyclooctyl-3-methoxybenzamide
1-ethyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(dimethylamino)-4-methyl-N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)pyrimidine-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl]pyridine-4-carboxamide
N-(adamantan-1-yl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(3R,5S)-5-[1-(3,4-dichlorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol
3-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-(4-cyanophenyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(1R,2R,4R)-N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-{5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-3-phenyl-1H-1,2,4-triazol-1-yl}pyridine
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
1-(propan-2-yl)-N-[3-(pyridin-3-yloxy)propyl]piperidine-4-carboxamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]propanamide
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-(morpholin-2-yl)ethan-1-one
methyl (2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-(2-methylpropanamido)pyrrolidine-2-carboxylate
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[(2R,3R)-1'-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
7-(2-hydroxypyridine-3-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}pyridine-2-carboxamide
4-[(1E)-3-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]prop-1-en-1-yl]-2-methoxyphenol
2-{1-cyclohexyl-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-5-phenoxyfuran-2-carboxamide
1-methyl-4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}imidazolidin-2-one
N-(furan-3-ylmethyl)-N-methyl-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
2-ethyl-5-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}pyrimidine
(3aR,6aR)-N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-methyl-3-(1-methyl-1H-pyrazol-5-yl)-N-[1-(pyridin-3-yl)pentyl]propanamide
3-({2-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-cyclopropyl-4-methoxy-2-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
N-(2-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}quinolin-6-yl)acetamide
4-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-1-phenylpiperazin-2-one
2-(2-chloro-6-fluorophenyl)-N-{2-[2-(2-methoxyethyl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}acetamide
2-[3-(3-fluorophenoxymethyl)-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
1-(prop-2-en-1-yl)-N-[2-(propan-2-yloxy)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(prop-2-en-1-yl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-propylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxamide