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1-cyclobutanecarbonyl-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
methyl 3-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(pyridin-3-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
3-[2-(3-methoxyphenyl)ethyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-N'-(5-methyl-1,2-oxazol-3-yl)ethanediamide
2-fluoro-N-[1-({[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
5-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-2,1,3-benzothiadiazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,1,3-trimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-methylpyrazin-2-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
1-cyclobutyl-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-(2-methoxyethyl)-1-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-{5-[(2,4-dioxoimidazolidin-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-ethyl-2-methylquinoline-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(6-ethylpyrimidin-4-yl)amino]pyrrolidin-2-one
5-[1-(2-methoxyacetyl)piperidine-3-carbonyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-ethyl-1,2-oxazole-3-carboxamide
(2S,4S)-1-methyl-4-[4-phenyl-5-(pyridin-2-yl)-1H-imidazol-1-yl]pyrrolidine-2-carboxylic acid
2-amino-4-(4-hydroxy-3-methoxyphenyl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-cyclopentyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[4-(oxolan-3-yloxy)phenyl]methyl}acetamide
2-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-phenoxy-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-(1-methylpiperidin-2-yl)-1-[4-(2-methylpyridin-4-yl)piperazin-1-yl]propan-1-one
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(5-methylfuran-2-yl)benzamide
1-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(2-methoxyphenyl)propan-1-one
2-(furan-2-yl)-5-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}pyrimidine
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-methyl-1,2-oxazole-5-carboxamide
(1R,2R,4R)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-({2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)cyclohexan-1-ol
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
4-[(4-fluorophenyl)sulfanyl]-6-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidin-2-amine
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridin-2-amine
1-(1-benzothiophene-5-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-(2-methoxyphenoxy)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
2-[1-(3-methylbutyl)-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
N-({5-[(1-ethyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-ethyl-3,4,7-trimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
4-[2-(piperidine-1-carbonyl)phenoxy]-1-(thiophen-3-ylmethyl)piperidine
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N,2-dimethyl-4-phenyl-N-(quinolin-5-ylmethyl)pyridine-3-carboxamide
1-(8-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}imidazo[1,2-a]pyridine-2-carbonyl)piperidine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
(4R,6S)-4-methyl-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-1,3-diazinane-2-thione
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{2-benzyl-1-methyl-7-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}propanamide
1-(1-benzofuran-2-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide