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(4aR,6R,8aS)-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-{[5-(3-cyclopropyl-1H-pyrazol-5-yl)-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
7-(5-chloropyridin-2-yl)-4-(3-fluorobenzoyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
4-[2-(1H-imidazol-2-yl)benzoyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
(3S,4R)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
ethyl 2-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]amino}acetate
1-(2-{[(3-methylphenyl)methyl]amino}-1-propyl-1H-1,3-benzodiazole-5-carbonyl)azetidin-3-ol
2-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-[(3,4-dimethoxyphenyl)methyl]acetamide
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-(naphthalen-2-ylmethyl)piperazin-2-one
3-hexyl-8-(2-hydroxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-benzylpiperidin-4-yl)-1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(1H-imidazol-1-yl)propanamide
(4aR,7aS)-1-(3-methylbutanoyl)-4-[(4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2E)-1-{3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]morpholin-4-yl}-3-phenylprop-2-en-1-one
N-(2-ethoxybutyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-[4-(2-chlorophenoxy)piperidin-1-yl]-9H-purin-2-amine
2-ethoxy-6-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
5-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-2-propylpyrimidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
N,2,3,6-tetramethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]quinoline-4-carboxamide
6-chloro-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
6-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
5-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-2-(pyrrolidin-1-yl)pyrimidine
N-[(2R,3R)-1'-(3,3-dimethylbutanoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
{2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}dimethylamine
N-{[7-(3-cyclohexylpropanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
(2R,6R)-4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3-[3-(trifluoromethyl)benzoyl]piperidine
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-(morpholin-4-yl)propan-1-one
N,3-dimethyl-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
ethyl 1-(5-benzamido-1-cyclopentyl-1H-1,3-benzodiazole-7-carbonyl)piperidine-2-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
(3S,4S)-4-(pyridin-2-yl)-1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
6-{4-[4-(cyclopropylcarbamoyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrazine-2-carboxamide
3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-[2-(pyridin-4-yl)ethyl]urea
3-(5-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-(furan-2-ylmethyl)-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carboxamide
N-{3-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}acetamide
1-methyl-2-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-1H-1,3-benzodiazole
N-butyl-N-[(4-fluorophenyl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-(1-{6-[4-(prop-2-en-1-yl)piperazin-1-yl]pyridine-3-carbonyl}piperidin-4-yl)morpholine
1-[(4-methoxy-3-methylphenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol