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2-methyl-5-phenyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-(oxolane-2-carbonyl)-1,4-diazepane
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}acetamide
4-[2-(2-methoxyethyl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-2-(2,5-dimethoxyphenyl)-N-(furan-2-ylmethyl)acetamide
2-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}-N-[4-(N-methylacetamido)phenyl]acetamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2,6-difluorophenyl)methyl]pyrrolidine-2-carboxylate
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(6-methylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(3-methylthiophen-2-yl)methyl]amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-(4-methylpiperidin-1-yl)propan-1-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
dimethyl(2-{[(3-methylthiophen-2-yl)methyl]({[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino}ethyl)amine
3-({1-[2-(2,3-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]propan-2-yl}oxy)pyridine
6-{[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(cyclopropylmethyl)-N-propylacetamide
N2,N2-dimethyl-N4-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
4-(3,4-dimethoxybenzoyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
methyl 4-{2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamido}butanoate
6-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]pyrimidin-4-amine
1-[(2-hydroxy-5-methoxyphenyl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)benzamide
4-[(2-methylphenyl)methyl]-1-(2-phenoxyacetyl)-1,4-diazepan-5-one
methyl 3-[(3,5-difluorophenyl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-N,N-dimethylaniline
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(naphthalen-2-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-N-methyl-1-oxo-N-(1H-pyrazol-3-ylmethyl)-2,3-dihydro-1H-isoindole-4-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(1-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
5-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(4aS,8aR)-2-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-decahydroisoquinoline
N-{2-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
3-[methyl({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl})amino]propane-1,2-diol
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(piperidin-1-yl)acetamide
6-fluoro-2-{[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)amino]methyl}quinolin-4-ol
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
4-phenyl-1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}azepane
1-{5-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]thiophen-2-yl}ethan-1-one
7-(3-phenylpropyl)-2-(prop-2-ene-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(ethylamino)-N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}pyrimidine-5-carboxamide
3-[1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-2-yl]propan-1-ol
{2-[4-(2,4-difluorobenzoyl)morpholin-2-yl]ethyl}dimethylamine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
3-(azocan-1-yl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
2-methyl-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(phenylamino)propan-1-one