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2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-ol
2-({4-methyl-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
1-[(5-acetylthiophen-3-yl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
ethyl 1-(2-methylpropyl)-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(4-methoxyphenyl)methyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
8-fluoro-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)quinoline-2-carboxamide
4,4,4-trifluoro-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-1-one
1-[4-(azepan-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]cyclopropane-1-carboxamide
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-(3-chlorophenyl)-4-[(2,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1,4-dioxan-2-ylmethyl)-3-[2-(4-fluorophenoxy)pyridin-3-yl]-1-methylurea
1-{2-[1-(3-chloro-2-methylphenyl)-3-(cyclopropylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
N-(2-methylpropyl)-5-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
N-[(2R,3R)-1'-(6-hydroxypyridine-3-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
3-methoxy-1-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]piperidine
N-[(4-fluorophenyl)methyl]-N-methyl-4-sulfamoylbenzamide
(4aS,7aR)-1-(1-methyl-1H-pyrazole-5-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(furan-2-yl)-2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]ethane-1,2-dione
1-methanesulfonyl-4-[2-(pyrrolidin-3-yl)benzoyl]-1,4-diazepane
2-[benzyl(methyl)amino]-N-(oxan-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
4-fluoro-N-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]benzamide
N-(3-aminopropyl)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carboxamide
5-{3-carbamoyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-7-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
5-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-methyl-8-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-2-(propan-2-yl)-1,3-benzoxazole
1,3-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-4-carboxamide
3-(furan-2-ylmethyl)-5-[1-(3-methylpentanoyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
4-fluoro-N-{2-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
N-{3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}-N-methylmethanesulfonamide
{1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]pyridin-2-amine
1-(2,4-dimethoxypyrimidin-5-yl)isoquinoline
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
N-(cyclopropylmethyl)-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-propylacetamide
1-[2-(1H-pyrazol-1-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
2-benzyl-N-(cyclobutylmethyl)-1-methyl-N-(oxolan-2-ylmethyl)-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
4-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-2-(trifluoromethyl)morpholine
3-(2-methoxyphenyl)-N-[2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
2-[(1-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperidin-4-yl)oxy]pyrimidine
3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.5]undecane
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}adamantan-1-amine
2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-1-methylazepane
8-(6-aminopyridine-3-carbonyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-benzylpiperazin-1-yl)-3-[1-(3-phenylpropyl)piperidin-3-yl]propan-1-one