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(3aS,6aS)-2-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(2R,3R,6R)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
methyl 5-({2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]acetamido}methyl)furan-2-carboxylate
2-{3-cyclopropyl-5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,2,4-triazol-1-yl}pyridine
1,3-dimethyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
{3-[(2,4-difluorophenyl)methyl]-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}methanol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-{[(3-methylthiophen-2-yl)methyl]amino}-N-[(3S)-2-oxoazepan-3-yl]benzamide
methyl[(5-methylfuran-2-yl)methyl]({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-ethoxy-1-(4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
5-(1-ethylpiperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
3-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]benzoic acid
4-methyl-3-(4-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)-4H-1,2,4-triazole
1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-3-phenylprop-2-yn-1-one
{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine
1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(1,3-benzoxazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
(1S,5R)-6-(2-methoxyethyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-(propan-2-yl)-1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-({8-[(4-chlorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-3-carboxamide
(2S)-2-{3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamido}-3-phenylpropanamide
ethyl 3-[(3-{[(4-phenylphenyl)formamido]methyl}piperidine-1-carbonyl)amino]propanoate
methyl 2-[8-(2,2-dimethylpropyl)-1-[2-(4-methoxyphenyl)ethyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]acetamide
(1S,5R)-3-(5-methoxy-1H-indole-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-benzyl-3-(pyridin-2-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-4-ylmethyl)-1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-cyclopropyl-4-methoxy-3-({1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
methyl 4-{5-chloro-2-[(pyridin-3-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
N-[5-(morpholin-4-yl)pentyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
N-[4-({4-[1-(2,3-dihydro-1H-inden-2-yl)-4-methyl-2,5-dioxoimidazolidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
8-(2,5-dimethylfuran-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-butyl-4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methylpyrimidin-4-amine
4-{1-[2-(propylsulfanyl)acetyl]piperidin-3-yl}benzoic acid
1-(4-hydroxyphenyl)-N,N-bis(1,3-oxazol-4-ylmethyl)-5-oxopyrrolidine-3-carboxamide
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-N,N-dimethylpyrrolidine-2-carboxamide
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(4-methoxyphenyl)-1-(3-methylbutyl)-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
(2E)-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methylpiperidin-4-amine
{4-[(5-propylfuran-2-yl)methyl]-1,4-oxazepan-6-yl}methanol
1-(carbamoylmethyl)-N-{[4-(dimethylsulfamoyl)phenyl]methyl}piperidine-3-carboxamide
1-[4-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
2-(2,5-dimethylfuran-3-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane