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ethyl 4-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methyl-1-[4-(oxan-2-ylmethoxy)phenyl]urea
ethyl 4-[6-(2H-1,3-benzodioxole-5-carbonyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
(4aS,8aR)-6-(3-methylbenzenesulfonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
N-benzyl-N-(cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-5-phenoxyfuran-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]acetamide
2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
3-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]isoquinoline
1-{[4-(cyclopentyloxy)phenyl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine
1-[2-(3-methylpyridin-4-yl)phenyl]ethan-1-one
5-(3-benzoylpiperidine-1-carbonyl)-3-chloro-1,2-dihydropyridin-2-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-cyclohexyl-4-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
9-methoxy-7-(2-methoxyphenyl)-4-(5-methylthiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-6-(2-methylpropyl)pyrimidine-4-carboxamide
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(piperidin-1-yl)propyl]amine
5-(2,3-dimethylphenoxy)-1-azabicyclo[3.2.1]octane
4-[2-(3-fluorophenyl)piperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)benzamide
N-[(1-cyclopentylpyrrolidin-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-3-amine
3-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2,5-thiadiazole
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-3-yl]methanol
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1-benzothiophene-2-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(4-fluorophenyl)-1H-indazol-1-yl]acetamide
2-{[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}-N,N-dimethylacetamide
3,4,7-trimethyl-2-[4-(thiophen-3-ylmethyl)piperazine-1-carbonyl]-1H-indole
2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
2-[4-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]-1-(pyrrolidin-1-yl)ethan-1-one
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-(dicyclopropylmethyl)-N-methylacetamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)acetamide
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-[1'-(1H-indazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)methanesulfonamide
1-cyclohexyl-4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(methylsulfanyl)propyl]amine
N4-(1H-imidazol-2-ylmethyl)-N4-methyl-7-(pyrimidin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N-(2-fluorophenyl)-3-hydroxypiperidine-1-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2,2-dimethylpropanamide
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-1-(2-methylpropyl)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2H-1,3-benzodioxol-5-yl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[4-(pyridin-3-yloxy)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidin-4-amine
5-ethyl-6-methyl-N4-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-2,4-diamine
7,8-dimethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]-4-(pyrrolidine-1-carbonyl)quinoline
N-[2-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
7-(1-ethylpiperidine-4-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide