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[(3R,4R)-1-(2,6-difluoro-3-methoxybenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-ethyl-2-{4-[2-(morpholin-4-yl)ethyl]piperazine-1-carbonyl}-1H-indole
1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-4-ol
6-oxo-1-(3-phenylpropyl)-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
N-(pyridin-2-ylmethyl)-3-{[1-(thiophene-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
1-(4-chlorophenyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]cyclobutane-1-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(2S)-1-hydroxypropan-2-yl]pyrimidine-5-carboxamide
2-[(quinoxalin-2-ylmethyl)(thiophen-3-ylmethyl)amino]butan-1-ol
(3R,5S)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-({[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(2-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-hydroxy-N-[(2-methoxyphenyl)methyl]-N-propylpyridine-3-carboxamide
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-[2-(pyridin-2-yl)pyrimidin-5-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-(butan-2-yl)-N-(pyridin-3-ylmethyl)acetamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(1H-1,2,4-triazol-1-yl)acetamide
3-{1-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-3-yl}benzoic acid
1-[2-(benzyloxy)ethyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
4-({1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl}oxy)pyridine
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propyl]piperidine-3-carboxamide
(4aR,8aR)-2-methanesulfonyl-7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-2,7-naphthyridin-4a-ol
2-(pyrazine-2-carbonyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyloxan-4-yl)methyl]propanamide
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1'-[(8-chloroquinolin-2-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}oxolane-2-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)propanamide
4-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)benzoic acid
7-(4-chlorophenyl)-2-(1-ethyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3R,4S)-4-cyclopropyl-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]pyrrolidin-3-yl]cyclohexanecarboxamide
5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-N-propylpyrimidin-2-amine
2-{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}ethan-1-ol
2-methyl-4-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenol
1-(carbamoylmethyl)-N-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidine-3-carboxamide
2-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-2-yl}pyridine
N-{2-[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
3-{[1-propyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
1-[(4-chlorophenyl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-({1-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}methyl)acetamide
N-[(3-methoxyphenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[3-({[1-(2-methoxyphenyl)propan-2-yl](methyl)amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
5-(2-fluorophenyl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1,2,4-triazin-3-amine
7-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2,7-diazaspiro[4.5]decane
3-[1-(cyclohexylmethyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
1-[(3-methoxyphenyl)methyl]-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine