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1-(1,3-benzothiazol-2-yl)-4-hydroxypiperidine-4-carboxylic acid
5-(4,6-dimethoxypyrimidin-2-yl)quinoline
2-[2-(1H-imidazol-4-yl)ethyl]-9-(3-methyl-1H-pyrazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1'-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-methyl-2-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}quinoline
2-{[2-(adamantan-1-yl)-4-hydroxypyrimidin-5-yl]formamido}-N-ethylpropanamide
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
6-(3,4-difluorobenzoyl)-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(6-methyl-2-propylpyrimidin-4-yl)-1λ6-thiomorpholine-1,1-dione
[1-(6-aminopyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methanol
methyl N-[2-(2-{[(3S)-3-fluoropyrrolidin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)-2-oxoethyl]carbamate
8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-methoxyphenyl)-3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-1-(3-methylbutyl)pyrrolidine-2,5-dione
4-benzoyl-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
(3R,9aR)-3-benzyl-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
5-{[2-(4-fluorophenyl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-(2-{1-[(3-chloro-5-fluorophenyl)methyl]piperidin-2-yl}ethyl)acetamide
1-(morpholin-4-yl)-3-[3-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
N-[(3R,4S)-4-(4-methoxyphenyl)-1-[2-(piperidin-1-yl)acetyl]pyrrolidin-3-yl]acetamide
2-fluoro-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5-sulfamoylbenzamide
1-(4-chlorophenyl)-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)cyclobutane-1-carboxamide
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-oxazolidin-2-one
1-[2-(4-methoxyphenyl)ethyl]-4-[(oxan-4-yl)amino]pyrrolidin-2-one
5-[1-(1-benzofuran-2-ylmethyl)pyrrolidin-2-yl]-3-methyl-1H-1,2,4-triazole
2,6-dimethyl-4-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}quinoline
4-[6-(methoxymethyl)pyrimidin-4-yl]-2-(trifluoromethyl)morpholine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-4-phenylbutan-1-one
2,3-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]quinoxaline-6-carboxamide
N-methyl-2-phenoxy-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-(3-fluorophenoxymethyl)-1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(methylamino)ethyl]benzamide
3-(cyclopropylsulfamoyl)-5-(6-methoxypyridin-3-yl)benzoic acid
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine-3-carboxamide
N-cyclopropyl-3-{5-[(6-methylpyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
5-fluoro-N2-[3-(furan-2-yl)propyl]-N4,N4-dimethylpyrimidine-2,4-diamine
N3-(1-benzothiophen-2-ylmethyl)-N5-cyclohexyl-1-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(thiophen-3-ylmethyl)piperazin-1-yl]ethan-1-one
3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1,3-benzothiazole-6-carboxamide
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-2,2-dimethyloxane-4-carboxamide
4-({5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)imidazolidin-2-one
2-(1H-indol-6-yl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
N-methyl-N-(3-methylbutyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetamide
(1R,5S,6R,7S)-3-methyl-6-[4-(pyridin-3-yl)piperazine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(butan-2-yl)-N3-[(3,4-difluorophenyl)methyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide