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4-{[4-(3-chloro-4-ethoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
N-[4-(morpholine-4-carbonyl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
methyl 3-{[4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-yl]amino}propanoate
(3S,5R)-1-[(4,5-dimethylfuran-2-yl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-4-(1H-pyrazol-1-yl)benzamide
N4-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-N6-(propan-2-yl)pyrimidine-4,6-diamine
{5-[1-(2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
2-(azocan-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
1-[(4aR,8aS)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
(3R,4R)-3-cyclobutyl-1-(3,5-difluoro-4-methoxybenzoyl)-4-methylpyrrolidin-3-ol
5-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4H,5H,6H,7H-thieno[3,2-c]pyridine
1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
1-(2H-1,3-benzodioxole-5-carbonyl)-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
4-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)thiomorpholine
N-({3-methyl-7-[4-(propan-2-yloxy)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-3-(1H-pyrazol-4-yl)benzamide
N-{4-[3,5-dimethyl-4-(2-oxopropyl)-1H-pyrazol-1-yl]-2-ethylphenyl}acetamide
1-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)-3-(morpholin-4-yl)propan-1-one
[(3R,4R)-1-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(4aR,7aS)-1-(pyridin-3-ylmethyl)-4-[2-(thiophen-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-1,2,3-triazole
N-[2-(3,4-dimethoxyphenyl)ethyl]-N,1-dimethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-3-(4-methylphenoxymethyl)piperidine
(1S,5R)-6-[(4-ethoxyphenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-[4-(4-propylpyrimidine-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
5-benzenesulfonamido-1-ethyl-2-methyl-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
2-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,5-dimethyl-1H-pyrrole
5-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-propylpyrimidine
7-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-1-(2-phenylphenyl)piperazin-2-one
N-cyclopentyl-1-(2-methylpropyl)-5-[2-(pyridin-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N2,N2-dimethyl-N4-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(2,3-dihydro-1H-isoindol-2-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
5-methyl-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-propoxyethan-1-one
2-(2,4-dimethylphenyl)-2-{methyl[3-(morpholin-4-yl)propyl]amino}acetic acid
(1R,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N,6-dimethyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
4-phenyl-N-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methyl)benzamide
(2E)-N-{[7-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
ethyl 3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
3-(4H-1,2,4-triazol-4-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}benzamide
N-butyl-3-methyl-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-3,4-dihydroquinazoline-7-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(5-methyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-ol
N-({4-hydroxy-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]azepan-4-yl}methyl)piperidine-1-carboxamide
N3-[(3-chlorophenyl)methyl]-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide