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N-methyl-5-{[methyl({2-methylpyrido[2,3-d]pyrimidin-4-yl})amino]methyl}pyrimidin-2-amine
(2R,6R)-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[3-(4-hydroxypiperidin-1-yl)propyl]-3,4-dihydroquinazolin-4-one
2-{1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidin-2-yl}ethan-1-ol
3-(4-fluorophenyl)-4-(2-phenylbenzoyl)piperazin-2-one
N-(1H-indol-3-yl)-1H-indazole-3-carboxamide
2-methyl-4-[3-(2-phenylethyl)-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl]pyridine
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]benzonitrile
N-({7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
2-methyl-1-[(5-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]pyrrolidine
3-(1-methylcyclopropyl)-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
N-[2-(benzyloxy)ethyl]-4-(piperidin-3-yl)benzamide
(4aS,8aR)-6-(3-methylpyrazin-2-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
N-{[8-(quinolin-7-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
3-[1-(2-amino-5-ethylpyrimidin-4-yl)piperidin-4-yl]-N-cyclopropylpropanamide
6-[(1R)-1-(4-methoxyphenyl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[2-(2-fluorophenyl)-1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
ethyl 1-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-4-(2-methoxyethyl)piperidine-4-carboxylate
N-(4-{4-[(2-hydroxybutyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
2-[1-(2-hydroxyethyl)-5-[4-methyl-2-(pyridin-3-yl)pyrimidin-5-yl]-1H-1,2,4-triazol-3-yl]acetamide
methyl 1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-4-carboxylate
(3S,4S)-N-(3,5-dichlorophenyl)-3,4-dihydroxypiperidine-1-carboxamide
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-phenylbutane-1,2-dione
8-(naphthalen-1-ylmethyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-[2-(1H-imidazol-1-yl)ethyl]-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
3-(2,4-dimethylbenzoyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(5-fluoro-1H-indole-2-carbonyl)-N,N-dimethylazepan-4-amine
5-chloro-2-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[4-(3-methylphenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(4-chlorophenyl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-methylbutan-1-one
1-[(3-chlorophenyl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-inden-1-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
methyl 3-{[1-(cyclopropylmethyl)-5-[4-(methylsulfanyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
6-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-2-methyl-1,3-benzothiazole
(3R,4S)-1-(5-methoxypyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-amine
N-(3-chloro-4-methylphenyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carboxamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
(4aS,8aR)-1-(2-methylpropyl)-6-(pyridin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-ethyl-1-(2-hydroxyethyl)-N-[2-(2-methylphenoxy)ethyl]piperidine-3-carboxamide
(3S,5R)-N3-[(3,5-dimethylphenyl)methyl]-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
N-(2-oxo-2-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)acetamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
3-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methoxy)pyridin-2-amine