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1-{4-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenyl}ethan-1-one
(1S,5R)-6-[(4-fluoro-2-methylphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)acetamide
7-(1-benzothiophene-2-sulfonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}butanamide
2-(5-{imidazo[2,1-b][1,3]thiazol-6-yl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)pyridine
2-(3-methylphenyl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(3R,4R)-4-ethyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3,4-diol
5-methoxy-3-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}methyl)-1H-indazole
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
4-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-5,6-dimethylpyrimidine
2,5-dioxo-6-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(2-{[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)amino}ethyl)piperidin-2-one
N-[1-(3,4-diethoxyphenyl)ethyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(methylsulfanyl)propanamide
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(4-fluorophenyl)piperidin-4-ol
2-(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(3-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-[(3S,4R)-1-[(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
3-benzyl-1-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indol-2-one
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
(2R,6S)-4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2,3-dihydro-1H-inden-2-yl}-2,6-dimethylmorpholine
N-[(2R,3R)-1'-(1H-imidazol-4-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
4-{3-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-ol
N-[1-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-methoxybenzamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(2-fluorophenyl)benzoyl]piperidine
1-[(2-chlorophenyl)methyl]-4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
(1S,5R)-6-benzyl-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{3-[4-(3-methylphenoxy)piperidin-1-yl]-3-oxopropyl}methanesulfonamide
1-{[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
4-{1-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyridine
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-(propan-2-yl)piperidin-4-yl]-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
1-[(4aR,8aS)-1-[2-(2,3,4-trifluorophenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
3-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5S,6R)-N-[2-(cyclohex-1-en-1-yl)ethyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N,N-diethyl-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-amine