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N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylbenzamide
(4aR,7aS)-1-ethyl-4-(morpholine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methyl-4-oxo-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)-1,4-dihydroquinoline-3-carboxamide
4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-[2-(diethylamino)ethyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-3,5-dimethoxybenzamide
N-[2-(3-chlorophenyl)ethyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(2-chlorophenyl)methyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
[2,4,6-trimethyl-3-({[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)phenyl]methyl acetate
ethyl 4-[4-(4-{[(2,3-difluorophenyl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
6-(difluoromethyl)-2-(3-{[(prop-2-en-1-yl)(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
9-(2-butoxyacetyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(2S,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
2-chloro-5-(5-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}furan-2-yl)benzoic acid
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
N-benzyl-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(thiophene-2-carbonyl)piperidine
1-{2-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-(cyclobutylmethyl)-3-hydroxy-3-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)piperidin-2-one
9-(3,4-dimethylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(4-methylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
5-methyl-N-(1,2-oxazol-3-ylmethyl)-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-{4-[4-(methylsulfanyl)benzoyl]morpholin-3-yl}-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]acetamide
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}benzamide
4-{[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
N-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]-4-methyl-1,3-thiazol-2-amine
N-{3-[methyl(phenyl)amino]propyl}oxane-4-carboxamide
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-[(4-chlorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-4-oxobutanamide
1-{2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]ethyl}piperidine-3-carboxamide
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
3-[2-(piperidin-2-yl)ethyl]-5-(pyridin-4-yl)phenol
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
N-cyclopentyl-2-{[3-(pyridin-3-yl)propyl]amino}propanamide
5-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(2-oxoimidazolidin-1-yl)benzamide
1-(cyclopropylmethyl)-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazine
(3R,4S)-4-cyclopropyl-1-(5-methoxyfuran-2-carbonyl)pyrrolidin-3-amine
4-[6-(2-methoxyphenyl)pyridazin-3-yl]-1-methylpiperazine-2-carboxylic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-cyclopropylacetamide
(1R,5S,8S)-3-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane