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5-(4-benzyl-3,5-dimethyl-1H-pyrazol-1-yl)pyrazin-2-amine
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(pyridin-2-yl)piperidin-4-ol
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
(3S,4S)-4-cyclopropyl-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
4-[4-(1H-pyrazol-5-yl)phenyl]benzamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-3-carboxylic acid
1-[7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
2-(4-fluorophenyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
2-(3-fluorophenyl)-N-{[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
1-(pyridin-3-yl)-2-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
(1S,5R)-6-methyl-3-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-{4,6-dimethyl-11-oxo-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-13-yl}phenoxy)acetic acid
(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-(hydroxymethyl)piperidin-3-ol
2-(naphthalen-1-ylmethyl)-4-(thiophene-3-carbonyl)morpholine
4-fluoro-3-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]benzene-1-sulfonamide
methyl 3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}benzoate
3-hydroxy-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
2-{[2-(cyclohexylmethyl)morpholin-4-yl]methyl}-5-methoxy-4H-pyran-4-one
(3R,4S)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-4-propylpyrrolidin-3-amine
6-chloro-2-[2-(methoxymethyl)pyrimidin-5-yl]-4-(piperidine-1-carbonyl)quinoline
methyl 4-(4-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(furan-3-ylformamido)methyl]benzoate
2-methyl-N-[6-methyl-2-oxo-4-(1-propyl-1H-imidazol-2-yl)-1,2,3,4-tetrahydroquinolin-7-yl]propanamide
(5S,9aS,9bS)-5-(2-chlorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-({[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
N-[(3,4-difluorophenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[4-(1H-pyrazol-3-yl)phenyl]methyl}piperidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-(2-phenylethyl)piperidin-3-amine
1-[2-(cyclohexylmethyl)morpholin-4-yl]-2-(2-hydroxyphenoxy)ethan-1-one
5-[(4-ethylpiperazin-1-yl)methyl]-N-(2-methoxyethyl)-1,2-oxazole-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[4-(5-ethyl-1,3-oxazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
(1H-1,3-benzodiazol-2-ylmethyl)(methyl){[5-(piperidin-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-({1-[3-(4-phenylphenyl)propanoyl]piperidin-4-yl}methyl)acetamide
4-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
N,N-dimethyl-4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
2-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
3-(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxane-2-carboxamide
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-2-(pyrrolidin-3-yl)acetamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine