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1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
(2S)-4-(methylsulfanyl)-2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)butan-1-ol
(2S,4S)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 4-{4-[({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)methyl]-5-methyl-1,3-oxazol-2-yl}benzoate
5-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-2,1,3-benzothiadiazole
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]quinoxalin-6-amine
4-(naphthalen-2-ylmethyl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
benzyl (1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[1-(4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
4-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}thiomorpholine
3-(2,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methoxybenzamide
4-[3-(2-methoxyphenyl)propanoyl]-1-methylpiperazine-2-carboxylic acid
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
8-[(2S)-2-amino-4-hydroxybutanoyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
N-({1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-3-yl}methyl)furan-2-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-3-[(2-hydroxypropyl)sulfamoyl]benzamide
2-(2-chloro-5-methylphenyl)-5-(methanesulfonylmethyl)pyridine
3-{[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-oxo-4H-chromene-2-carboxamide
4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-ethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
2-{4-[2-(trifluoromethoxy)phenyl]phenyl}acetamide
3-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-2-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
N-[4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]acetamide
3-(3-fluorophenyl)-3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-(naphthalen-1-yl)ethan-1-one
2-acetamido-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)acetamide
3-(propan-2-yl)-1-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidin-3-yl)methyl]urea
2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
2-[(5-chlorothiophen-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
5-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
({4-[2-(dimethylamino)ethoxy]phenyl}methyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
4-{[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]methyl}benzoic acid
(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl](oxolan-3-ylmethyl)amine
2-(cyclopropylmethyl)-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
1-benzyl-8-(cyclohex-3-en-1-ylmethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione