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4-[(4-methylphenyl)sulfanyl]-1-(1H-pyrrole-2-carbonyl)piperidine
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
3-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-(1-{6-[(3-hydroxy-2,2-dimethylpropyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
2-[3-(cyclopropylcarbamoyl)phenyl]-2-(thiomorpholin-4-yl)acetic acid
2-[5-(4-chloro-2-methoxyphenyl)-1-cyclohexyl-1H-1,2,4-triazol-3-yl]acetamide
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-benzoyl-4-(1-ethyl-3-methylpiperidine-3-carbonyl)piperazine
2-methyl-N-[(3-methylpyridin-2-yl)methyl]-N-(propan-2-yl)thieno[2,3-d]pyrimidin-4-amine
3-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
N-[4-(3-methoxyphenyl)phenyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxamide
{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]quinolin-3-yl}methanol
1-phenoxy-2-[4-(quinolin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-(dimethyl-1,2-oxazol-4-yl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
4-(4-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)-2-methylbut-3-yn-2-ol
N-[2-(2-fluorophenyl)-1-[1-(2-hydroxyethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
2-[4-(9-methyl-9H-carbazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-4-(1H-pyrazol-1-yl)butan-2-ol
6-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-[1-(cyclohexylmethyl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
2,6-dimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-[(4-ethylphenyl)methyl]-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
3-[4-(2,6-dimethylpyridine-4-carbonyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
N-methyl-5-[(2-methylpiperidin-1-yl)methyl]-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-ethyl-N4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-methylpyrimidine-2,4-diamine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-[(3-methylquinoxalin-2-yl)methyl]azepan-3-amine
(4aR,7aS)-1-benzyl-4-(3-methoxypropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[cyclohexyl(methyl)amino]-3-[2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
1-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[(2-chlorophenyl)methyl]-N-[2-(pyrazin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl){[4-(methylsulfanyl)phenyl]methyl}amine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
1-cyclopentyl-N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-6-oxopiperidine-3-carboxamide
10-methoxy-5-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
8-{[2-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[(5-cyclohexylthiophen-2-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(2-fluorophenyl)methyl]piperazin-2-yl)ethan-1-ol
methyl 2-[1-(2-methoxyethyl)-8-({4-[methyl(phenyl)amino]phenyl}methyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(1S,6R)-N-benzyl-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-sulfonamide
{3-[(3-chlorophenyl)methyl]-1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl}methanol
N3-(furan-2-ylmethyl)-N5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 1-(1-methylpiperidine-2-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[(3S,4R)-1-(5-chloropyridine-2-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(1S,6R)-9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
1-cyclohexyl-5-(2-ethoxyethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole