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2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]ethan-1-one
N-methyl-N-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}oxolan-3-amine
2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1,3-benzothiazole
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]urea
1-(4-fluorophenyl)-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyrrolidin-2-one
N-{2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}acetamide
2-(4-{[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
3-{[4-(3,4-difluorobenzoyl)piperidin-1-yl]methyl}piperidin-3-ol
1-(4-chlorophenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
2-{4-[(4-ethylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-methyl-4-(3-{4-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
3,5-dihydroxy-4-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-methanesulfonyl-1,4-diazepane
2-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
1-(cyclohexylmethyl)-N-ethyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-[4-(thiophen-2-ylmethyl)morpholin-3-yl]acetamide
N-[2-(3-methoxyphenyl)-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)ethyl]-N-methylcyclopropanecarboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
8-(4,6-dimethoxypyrimidin-2-yl)quinoline
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(3-hydroxypropyl)-1-methylpyrrolidine-3-carboxamide
2-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrido[2,3-d]pyrimidin-4-amine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
(1R,2R)-2-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)cyclohexan-1-ol
4-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1H-pyrrole-2-carbonitrile
N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}thiophene-2-carboxamide
N-(3,3-diphenylpropyl)-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-2-(trifluoromethyl)morpholine
3-(furan-2-ylmethyl)-1-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-1-methylurea
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-(2H-1,3-benzodioxol-5-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}piperidin-4-amine
N-(2-methoxyethyl)-4-(N-methylmethanesulfonamido)-N-[(4-methylphenyl)methyl]benzamide
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
N-[2-(methylsulfanyl)phenyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
2-(1-benzothiophen-2-ylmethyl)-4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(1R,3S)-3-ethoxy-7-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-7-azaspiro[3.5]nonan-1-ol
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-[(3,4-dimethoxyphenyl)methyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazol-3-yl}-N-methylformamido)-N-methylpropanamide
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
6-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
(1S,5R)-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(2-hydroxyethyl)piperazin-1-yl]-N-[4-methyl-3-(propan-2-yl)phenyl]piperidine-1-carboxamide
(1-benzothiophen-5-ylmethyl)[1-(4-methylpiperazin-1-yl)propan-2-yl]amine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}ethan-1-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
(2S)-2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-4-(methylsulfanyl)butan-1-ol