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N-ethyl-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-methylprop-2-en-1-yl)propanamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-(5-acetylthiophen-3-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
N-(1-cyanocyclohexyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
[(1-{[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
5-({methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}methyl)pyrimidin-2-amine
N-(3-acetylphenyl)-3-[(2-fluorophenyl)methyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridine-6-carboxamide
1-(3-{[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-indol-1-yl)ethan-1-one
2-[(4-chlorophenyl)methyl]-4-[4-(2-ethylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[(3,4-difluorophenyl)methyl]-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
3-{5-[(2,2,2-trifluoro-1-phenylethoxy)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
3-[5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-cyclopropyl-N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-4-(trifluoromethoxy)benzene-1-sulfonamide
(3S)-3-ethyl-4-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)morpholine
N-methyl-2-{4-[(E)-2-phenylethenyl]-1H-pyrazol-1-yl}acetamide
2-(4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenoxy)acetic acid
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-methyl-6-oxo-N-[2-(piperidin-1-yl)ethyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(pyridin-3-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(2-methylpropyl)-5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-1,2,4-triazole
1-(dimethylamino)-3-{4-methoxy-2-[({[1-(piperidin-1-yl)cyclopentyl]methyl}amino)methyl]phenoxy}propan-2-ol
1-(4-methoxybenzoyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
1-{5-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
6-methyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(7-chloro-4-{[(4-fluorophenyl)methyl]amino}quinazolin-2-yl)methyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(3-methoxybenzoyl)piperidine
[1-(3-fluorobenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N4-methyl-6-(morpholin-4-yl)-N4-[2-(1H-pyrazol-4-yl)ethyl]pyrimidine-2,4-diamine
2-(2,4-dichlorophenoxy)-N-(1,4-dioxan-2-ylmethyl)acetamide
(1S,2S)-2-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)cyclohexan-1-ol
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(4-methylphenyl)propan-1-one
4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-imidazol-2-yl]pyridine
4-{5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}pyridine
4-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-ol
N-{3-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]phenyl}acetamide
1-[2-(morpholin-4-yl)ethyl]-3-[3-(1,3-oxazol-5-yl)phenyl]urea
5-({3-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
[(3S,5R)-1-[6-(dimethylamino)pyrimidin-4-yl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
methyl 2-({3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}formamido)-4-(methylsulfanyl)butanoate
4-(4-chlorophenyl)-1-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}butan-1-one
[(2-fluorophenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]cyclopentanecarboxamide
N-[(2R,3R)-1'-[2-(2-fluorophenyl)acetyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-butoxy-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(3-methyl-1H-pyrazole-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane