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(2R,3S,6R)-3-(3-methoxyphenyl)-5-(morpholine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
dimethyl({[4-methyl-5-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-3-(3-hydroxy-3-methylbutyl)benzamide
2,6-dimethyl-N-[2-(1,3-thiazol-2-yl)ethyl]quinoline-4-carboxamide
1-(3-fluoro-2-methoxybenzoyl)-N,N-dimethylazepan-4-amine
4-methoxy-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
4-(1H-pyrazol-1-yl)-1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidine-4-carboxylic acid
7-(4-ethyl-5-methylthiophene-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(3,4-dimethoxyphenyl)-7-methyl-3-[(4-methylpiperazin-1-yl)methyl]quinoline
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-[(phenylsulfanyl)methyl]furan-2-carboxamide
2-(3-acetyl-1H-pyrazol-1-yl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-phenoxypropan-1-one
N-[(3-chlorophenyl)methyl]-2-(1-ethylpiperidin-4-yl)-N-methylacetamide
4-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2,3-dihydro-1H-imidazol-2-one
6,7-dimethoxy-3-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(1-benzofuran-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-benzyl-3-(2-methoxyethyl)-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
N-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)propan-2-yl]thiophene-2-carboxamide
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylfuran-3-carboxamide
3-(dimethylsulfamoyl)-5-({[2-(furan-2-yl)phenyl]methyl}amino)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
1-methyl-4-phenyl-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(4-hydroxyphenyl)ethyl]propanamide
4-(3,4-dichlorobenzoyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-(dimethylamino)-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethan-1-one
1-{[4-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
3-({2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-4-methyl-4H-1,2,4-triazole
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl][(2-methyl-1H-imidazol-4-yl)methyl]amine
3-{2-oxo-2-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethyl}-1,2,3-oxadiazol-3-ium-5-olate
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(6-methoxypyridin-3-yl)methyl]morpholine-2-carboxamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
(3aS,6aR)-5-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl 1-[2-(dimethylamino)ethyl]-5-[4-(4-methoxyphenyl)butan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
6-ethyl-N-[3-(trimethyl-1H-pyrazol-1-yl)propyl]pyrimidin-4-amine
1-{5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}azetidin-3-ol
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(5-methylthiophen-2-yl)methyl]benzamide
1-(4-fluorophenyl)-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
(2S,4R)-N-ethyl-1-(naphthalen-2-ylmethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
3-chloro-5-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N,3-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-propylthiophene-3-carboxamide
4-(5-ethoxyfuran-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-{4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenoxy}ethyl)acetamide
methyl 1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine-4-carboxylate
(2S)-2-{[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}propanamide