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6-oxo-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
2-(1-ethyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(3-chlorophenyl)methyl]-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-cyclopentanecarbonyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-[1-(3-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propan-1-ol
6-[2-(2-chlorophenyl)acetyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
5-methoxy-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-4-oxo-4H-pyran-2-carboxamide
5-({4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-(3-ethoxypropyl)-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-{1-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
(2R)-2-acetamido-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}butanamide
2,6-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)pyrimidine-4-carboxamide
2-[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1R,2R,6S,7S)-4-(3-methyl-1-benzothiophene-2-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
5-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
3,5-dimethyl-N-{2-[2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1,2-oxazole-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-oxopyrrolidin-1-yl)propanamide
2-(2,3-difluoro-4-methoxyphenyl)-1-[(4-methoxyphenyl)methyl]-1H-imidazole
1-[2-(butan-2-yloxy)phenyl]-3-[(1-propyl-1H-imidazol-2-yl)methyl]urea
N-ethyl-5-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
2-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)pyrimidine-5-carboxamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpyrrolidin-3-ol
9-(3,4-difluorobenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}urea
3-[2-(furan-2-ylmethoxy)phenyl]-1-methyl-1-(thian-4-yl)urea
4-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-methylbutanamide
3-({[(3,5-difluoro-4-methoxyphenyl)methyl]amino}methyl)piperidin-3-ol
N4-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-N2,6-dimethylpyrimidine-2,4-diamine
(2R,6R)-4-(2-amino-2-methylpropanoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(3-chlorophenyl)-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
methyl 3-benzamido-5-{[(3-fluorophenyl)methyl]amino}-1-(furan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
9-(2-methyl-1,3-thiazole-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-methylthiophen-2-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(prop-2-en-1-yl)propanamide
(2S,4R)-4-amino-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
2-(2-methoxy-5-methylphenyl)-2-[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]acetic acid
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-2-carboxamide
1-methyl-9-(prop-2-en-1-yl)-4-[2-(2H-1,2,3-triazol-2-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1-tert-butyl-1H-pyrazol-4-yl)-N-ethyl-N,8-dimethylquinoline-4-carboxamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[(2S,4R,6R)-2-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-6-(propan-2-yl)oxan-4-yl]acetamide
ethyl 2-{1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazol-3-yl]-N-methylformamido}acetate
N-(6-chloropyridin-3-yl)-4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-amino-N-(3-phenylpropyl)-N-(propan-2-yl)cyclopropane-1-carboxamide
(3S,4R)-N-(2,5-dimethylphenyl)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carboxamide