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{3-[(3-methyl-1,2-oxazol-5-yl)methyl]-9-[(4-methyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
2-{[4-(3-chlorophenyl)-5-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-methyl-N-[2-(2-methylphenyl)-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide
N-[2-(1-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}piperidin-2-yl)ethyl]acetamide
4-[1-(4-fluorophenyl)propan-2-yl]-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,2-dimethyl-1-benzofuran-5-carboxamide
methyl 4-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]butanoate
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
3-(1H-imidazol-2-yl)-1-(5-phenoxyfuran-2-carbonyl)piperidine
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-(4-fluorophenyl)pyrrolidine-1-carboxamide
3-(2-fluorophenyl)-3-[(2,6,8-trimethylquinolin-4-yl)formamido]propanoic acid
(2-{2-[1-(8-chloroquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
2-{2-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
N-({7-[2-(2-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-methyl-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-methyl-1'-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
1-(1,3-oxazole-5-carbonyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
(3aR,6aR)-2-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-methoxy-3-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
6-(hydroxymethyl)-N-[2-(3-methoxyphenyl)phenyl]-1,4-oxazepane-4-carboxamide
5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole
2-[(2-phenylethyl)(pyridin-2-ylmethyl)amino]butan-1-ol
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(morpholin-4-yl)butan-1-one
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)thiomorpholine
2-(4-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
2-{[(2-fluorophenyl)methyl](methyl)amino}-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-(oxan-2-yl)furan-2-yl]methyl}amine
ethyl 1-benzyl-5-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-(benzyloxy)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(3S,4S)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
(2S,4S)-4-amino-1-(2-amino-4-phenylpyrimidine-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
ethyl 4-{6-[4-(1H-imidazol-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(4-methyl-1H-imidazole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(4-{2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}piperidin-1-yl)pyrazine
N-{1-[1-(2,5-dimethoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
5-chloro-3-methyl-N-[(3R)-pyrrolidin-3-yl]-1H-indole-2-carboxamide
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-amido)cyclopentane-1-carboxylic acid