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1-(carbamoylcarbonyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-[3-(dimethylamino)pyrrolidine-1-carbonyl]-N-[(3-methyloxetan-3-yl)methyl]benzene-1-sulfonamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[1-(2-phenylethyl)piperidin-4-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3S,4S)-4-(3-methoxyphenyl)-1-(1H-1,2,4-triazole-5-carbonyl)piperidin-3-ol
N-[3-hydroxy-1-(4-methylphenyl)propyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-amino-4-[2-(propan-2-yl)pyrimidin-5-yl]-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
5-benzyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-(1-phenylbutyl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
2-methoxy-4-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(piperidin-1-yl)pyrimidine
2-cyclopropyl-9-[2-(4-fluoro-2-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-N'-[2-(morpholin-4-yl)ethyl]butanediamide
N-methyl-4-{1-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-imidazol-2-yl}benzene-1-sulfonamide
(1S,6R)-3-methyl-4-oxo-N-(6-phenoxypyridin-3-yl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
5-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(4-ethylpiperazin-1-yl)ethan-1-one
5-{1-[(3,4-dimethoxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
methyl(1,2-oxazol-3-ylmethyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
(2E)-N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-3-(3,4-dimethoxyphenyl)-N-(pyridin-3-ylmethyl)prop-2-enamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-N-methylpiperidine-2-carboxamide
2-(2-chloro-4-fluorophenyl)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}spiro[2.2]pentane-1-carboxamide
(2S,4S,5R)-4-[(1,3-dihydroxypropan-2-yl)carbamoyl]-2-ethyl-5-(4-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
3,3-dimethyl-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
(2S,4S)-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-methyl-2-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)acetamide
3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4-methyl-1,2,5-oxadiazole
2-methyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2,4-triazin-3-amine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(propan-2-yl)pyrimidine-4-carboxamide
N,N-dimethyl-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine-1-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-{[2-(1-benzyl-1H-pyrazol-4-yl)phenyl]methyl}propanamide
N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
2-{4-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]phenyl}ethan-1-amine
2-[3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]acetic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
3-[(3R,4S)-1-[(5-chlorothiophen-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
5-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-2-(thiophen-2-yl)pyrimidine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylacetamide
N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
N-{3-[(dimethylsulfamoyl)amino]phenyl}azetidine-1-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
(2S,4S)-N-[(5-fluoro-2-methylphenyl)methyl]-4-(3-methoxybenzamido)-1-methylpyrrolidine-2-carboxamide