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1-[(4-fluoro-2-methoxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[2-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
2,5-dimethyl-N-[2-(5-methyl-4-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-3-carboxamide
methyl 2-[(1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]phenyl}piperidin-4-yl)amino]acetate
methyl 3-[(2-methoxyphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(cyclopentylsulfamoyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
9-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
3-{[4-(pyridin-4-yloxy)piperidin-1-yl]methyl}pyrrolidin-3-ol
N-[1-(7-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]acetamide
2-{1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}ethan-1-amine
3-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazol-5-amine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-5-methyl-1,2-oxazole-4-carboxamide
4-({4-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)benzoic acid
1-(2-ethylbenzoyl)-2-(pyrrolidine-1-carbonyl)piperazine
N-[2-(2-fluorophenoxy)ethyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
2-methoxy-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-{4-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)acetic acid
N-({7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3,5-dimethoxy-2-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}benzoic acid
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methylpentane-1,4-dione
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
N-(furan-2-ylmethyl)-3-[2-(3-methoxyphenyl)azetidin-1-yl]propanamide
2-methyl-4-{4-[3-(pyridin-3-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
3-methyl-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
9-(2-propoxyacetyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-[(diethylcarbamoyl)methyl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-amino-1-{3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-N-methylpyrrolidine-2-carboxamide
3-butanamido-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylbenzamide
dimethyl({[4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,4-oxazepan-6-yl]methyl})amine
1-(5-fluoropyridin-3-yl)-3-(thiolan-3-yl)urea
N-cyclopropyl-1-[(1s,4s)-4-{[(3-methoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
6-(3-ethoxy-2-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2-(cyclohexylmethyl)-4-(4-methyl-1,3-oxazole-5-carbonyl)morpholine
4-hydroxy-2-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}quinoline-6-carboxamide
2-{[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]sulfanyl}-6-methyl-3,4-dihydropyrimidin-4-one
3-[({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]pyrrolidin-3-ol
5-ethyl-N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
{4-[(3-ethoxy-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
N-cyclopropyl-1-[1-(1H-indazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N,N-dimethyl-6-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxamide
(2S,4S)-4-[(adamantan-2-yl)amino]-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-(3,4-difluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide