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N-({8-[(3-ethoxy-4-hydroxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methylpropanamide
N-(1-benzothiophen-2-ylmethyl)-2-cyclobutyl-5-(2-methoxyacetamido)-N,1-dimethyl-1H-1,3-benzodiazole-7-carboxamide
2-(2-{[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-benzyl-5-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)pyrimidin-2-amine
N-[1-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-phenoxyacetamide
2-{4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
N-[2-(3-chlorophenyl)ethyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
5-[(2-chlorophenyl)methyl]-5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
{2-[1-(2-methoxybenzenesulfonyl)piperidin-2-yl]ethyl}dimethylamine
N-(4-methoxyphenyl)-1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-amine
N-[4-(4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
N-[2-(2-fluorophenyl)ethyl]-5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
1-(cyclopropylmethyl)-5-(6-oxo-1,6-dihydropyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
4-hydroxy-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-cyclopentyl-3-(3-fluorophenyl)pyrrolidine-2,5-dione
N-(5-chloro-2-methoxyphenyl)-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
9-[(3-methylthiophen-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
ethyl 1-(2-methoxyacetyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
1-ethyl-4-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
1-[(2,3-difluorophenyl)methyl]-4-(1-methanesulfonylpyrrolidin-3-yl)piperidine
4-({[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2,6-dimethoxyphenol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)oxane-4-carboxamide
methyl 5-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-[(1,2,3,4-tetrahydronaphthalen-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-benzyl-5-methanesulfonamido-N,2-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
4-[(furan-2-ylmethyl)amino]-N-(1-methoxypropan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
14-(6-ethoxypyridin-3-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-(azetidine-1-carbonyl)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]benzene-1-sulfonamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propanamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-(adamantan-1-yl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
3-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-(propan-2-yl)-1,2-oxazole
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperazine-1-carboxamide
2-methyl-N-(oxolan-3-yl)-1-benzofuran-5-carboxamide
2-(4-methylpentyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]morpholine
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
1-[2-(dimethylamino)ethyl]-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]piperidin-2-one
4-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[3-(pyridin-2-yl)propyl]benzamide
4-{1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-3-yl}benzoic acid
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine