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8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-[2-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetic acid
N-[1-(4-methylphenyl)ethyl]-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}acetamide
methyl 5-(cyclopentylamino)-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-[(2-methylphenyl)methyl]-1-(oxolan-2-ylmethyl)urea
(3R,5S)-N-cyclopentyl-1-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
4-{[(4-methylphenyl)amino]methyl}-N-[4-(pyrrolidin-1-yl)butyl]benzamide
3-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1-(thiophen-2-yl)urea
9-[(3-fluoro-2-methylphenyl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(1-methyl-1H-pyrazol-4-yl)propyl]amine
3-(2-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-2-oxoethyl)-3-(2-methylphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
(3R,7S,8aS)-7-[(1,3-benzothiazol-2-ylmethyl)amino]-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]but-3-en-1-one
2-methyl-1-[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)azetidin-3-yl]piperidine
3-(1H-1,3-benzodiazol-2-yl)-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
(2S,4R)-1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-N-[2-(3-chlorophenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
5-fluoro-2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-2-yl}-1H-1,3-benzodiazole
methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})(quinoxalin-6-ylmethyl)amine
N-(1-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-methylfuran-3-carboxamide
1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(1H-pyrazol-1-yl)butan-1-one
2-(4-hydroxyphenyl)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(thian-4-yl)piperazine
5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(pyrazin-2-yl)propanamide
5-(3-fluorophenoxymethyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
N-ethyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pentan-3-yl)acetamide
4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-[(3-fluorophenyl)methyl]-4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-(1H-pyrazol-3-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}benzamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-ethyl-N-methyl-6-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
methyl 3-(4-tert-butylbenzoyl)-9-[3-(dimethylamino)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{1'-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3-(4-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
3-(3-hydroxy-3-methylbutyl)-N-[4-(hydroxymethyl)oxan-4-yl]benzamide
N-[2-(adamantan-1-yl)propan-2-yl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(3-chlorophenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
8-(4-methylpiperidine-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S)-1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxy-3-phenylpropan-1-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)ethan-1-one
2-methyl-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-3-(1H-pyrazol-1-yl)propanamide
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[2-(pyridin-4-yl)ethyl]pyrrolidine-3-carboxamide
4-(1H-1,3-benzodiazol-2-ylmethyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
2-[5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N4-methyl-N6-(propan-2-yl)-N4-(1H-pyrazol-5-ylmethyl)pyrimidine-2,4,6-triamine
1-cyclohexyl-4-(5-phenyl-1,2-oxazole-3-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-methoxy-N-[1-(2-phenylethyl)-7-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]acetamide