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N-[2-(dimethylamino)ethyl]-5-ethyl-N,2,3-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
4-({5-[5-(methoxymethyl)furan-2-yl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
3-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)-1-methylpyrrolidine-2,5-dione
5-[2-(2-chloro-6-fluorophenyl)acetyl]-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
11-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
4-methoxy-N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
N5-[2-(3-chlorophenyl)ethyl]-N3-ethyl-1-(2-methoxyethyl)-N3-(2-methylprop-2-en-1-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclooctyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-{[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzoic acid
ethyl 1-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-1-propylpiperidin-4-amine
2-{9-[2-(methylsulfanyl)propanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-[2-(4-fluorophenyl)ethyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(morpholin-4-yl)ethyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
3-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
2-(butylsulfanyl)-5-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}pyrimidine
4-(2,6-dimethylpyridin-3-yl)-2-{pyrazolo[1,5-a]pyridin-7-yl}pyrimidine
2-{4-[(6-ethoxyquinolin-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-[4-(furan-2-yl)butan-2-yl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
1-(4-{[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}thiophen-2-yl)ethan-1-one
2-{4-[4-(benzyloxy)butanoyl]-2-oxopiperazin-1-yl}benzonitrile
N-[4-(2-amino-3-cyano-6-ethyl-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl)phenyl]acetamide
2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N-methylethane-1-sulfonamide
N-(4-{[1-(butan-2-yl)-1H-pyrazol-5-yl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
3-{[3-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-N-(1,2-oxazol-3-ylmethyl)benzamide
5-{[(2R,3R)-2-methoxy-3-(2-methylpropanamido)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylpropanamide
2-ethyl-9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidine-4-carboxylate
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({4-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)methylamine
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(4-fluorophenyl)piperidin-4-yl]acetamide
4-methoxy-2-{[8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
8-(cyclohexylmethyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]acetamide
N-[2-(pyrazin-2-yl)ethyl]-2-(thiophen-2-yl)acetamide
(4aS,8aR)-6-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-(morpholine-4-carbonyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyridin-2-amine
N-cyclopropyl-2-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}oxy)-4-methoxybenzamide
N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-2-{4-[4-(trifluoromethyl)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
3-(1-hydroxy-3-methylbutan-2-yl)-5-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N-[2-(azepan-1-yl)-2-phenylethyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]ethane-1-sulfonamide
N-[(4-fluorophenyl)methyl]-3-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]propanamide
methyl 4-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazole-3-carboxylate