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(2R,3R,6R)-5-(furan-2-carbonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methoxy-N-[1-methyl-7-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazol-5-yl]acetamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-4-phenylbutane-1,4-dione
2-cyclopentyl-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
3-{5-[2-(ethylsulfanyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-{1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-(2-{7-[(2-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-(3-methylphenyl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
4-(5-chloro-2-methoxybenzenesulfonyl)-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-methanesulfonylpiperidin-4-yl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
7-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(2H-1,3-benzodioxol-4-ylmethyl)[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
6-[methyl(propan-2-yl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-{[1-(thiophene-2-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
2-ethoxy-6-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)phenol
5-(2-methylphenyl)-4-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-2-(pyridin-3-yl)pyrimidine
N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-1,4-diazepane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-(5-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
4-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
(2E)-N-({7-[3-(4-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
N-benzyl-2-[6-hydroxy-4-(piperidin-4-yl)-1,4-diazepan-1-yl]acetamide
1-cyclopentanecarbonyl-N-[(2,3,4-trifluorophenyl)methyl]piperidine-4-carboxamide
4'-(2,2-dimethylpropyl)-1-propyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
N-(2-methoxy-2-methylpropyl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
7-methoxy-N,N-dimethyl-2-(2-phenylpyrimidin-5-yl)quinoline-4-carboxamide
2-methoxy-3-[6-(propan-2-yl)pyrimidin-4-yl]quinoline
1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-N-methylpiperidine-3-carboxamide
N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(methylamino)benzamide
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
5-(6-methyl-5-{[2-(thiophen-3-yl)acetamido]methyl}-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)-2,1,3-benzoxadiazol-1-ium-1-olate
8-fluoro-2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,4-dihydroquinolin-4-one
2-methanesulfonyl-N-(2-phenylethyl)-N-(propan-2-yl)acetamide
1-(2-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-5-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
1-[3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzoyl]azepane
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
5-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-one
[(1-{1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
N-(1H-indol-6-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 1-[(3R,5S)-1-(2-ethylbutyl)-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 3-(1-benzofuran-2-ylmethyl)-9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(cycloheptylcarbamoyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-acetyl-N-(1,2-oxazol-3-ylmethyl)benzamide