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(1R,3S)-3-(2-aminoethoxy)-7-[(3-methylquinoxalin-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
8-cyclobutyl-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(2,4-difluoro-3-methoxybenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[3-(2-methylphenyl)phenyl]-N-[2-(pyridin-4-yl)ethyl]piperidin-4-amine
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-cyclohexyl-3-[(1-methyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]propanamide
methyl 4-[4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazine-1-carboxylate
9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-(dimethylamino)-7-(3-methyl-1-benzothiophene-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4'-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
(2S,4R)-1-(1-benzothiophen-2-ylmethyl)-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
8-[(4-chlorophenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}amine
3-amino-1-(3-phenylpropyl)pyrrolidine-3-carboxylic acid
3-(1H-1,3-benzodiazol-2-yl)-1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]propan-1-one
1-[4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
1-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
2-(phenylsulfanyl)-N-[1-({[1-(thiophen-3-yl)propan-2-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}propanamide
2-({4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}sulfanyl)ethan-1-ol
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[(3-methylthiophen-2-yl)methyl]amine
1-{1'-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-cyclopentanecarbonyl-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-{2-[4-(1-benzothiophen-2-ylmethyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-(4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
4-(4-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-yl}phenyl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
2-(5-acetylthiophen-3-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethan-1-one
3-(3-hydroxyquinoxalin-2-yl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}propanamide
2-[1-(5-methyl-4-{methyl[2-(4-methylphenoxy)ethyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperidin-2-yl]ethan-1-ol
5-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylfuran-3-carboxamide
3-[4-(furan-2-yl)butan-2-yl]-1-(3-methanesulfonamido-4-methoxyphenyl)urea
3-{[5-(ethylsulfanyl)-1,3,4-oxadiazol-2-yl]methyl}-3,4-dihydroquinazolin-4-one
2-[5-(2,3-dihydro-1-benzofuran-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-2,5-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
(4aS,7aR)-1-(1H-1,3-benzodiazole-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(4-hydroxyphenyl)-5-[1-(2-methylpropanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[2-(2,4-dichlorophenyl)ethyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2-(2,2-dimethyloxan-4-yl)-1-(3-ethoxypropyl)-1H-imidazole
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methylpyrimidine
1-(furan-2-carbonyl)-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-1,4-diazepane
3-chloro-6-{3-[2-(dimethylcarbamoyl)ethyl]piperidin-1-yl}pyridine-2-carboxylic acid
3-(5-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid