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N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-N-propyl-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-2-yl)ethan-1-one
4-(5-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
N,4-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazole-5-carboxamide
2-methoxy-5-{[4-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
2-[benzyl(methyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
4-(dimethyl-1,2-oxazol-4-yl)-3-[3-(morpholin-4-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-fluoro-3-methyl-2-{[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-indole
N-[2-(1H-imidazol-4-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}bis(prop-2-en-1-yl)amine
N-[4-(methylsulfanyl)phenyl]-6-[(2,4,5-trimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(dimethylamino)ethyl]-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
4-(dimethyl-1,2-oxazol-4-yl)-N,6-dimethyl-N-(2-methylpropyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[2-(4-{[2-(2,5-dimethoxyphenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
{3-[(4-fluorophenyl)methyl]-1-(pyrazine-2-carbonyl)piperidin-3-yl}methanol
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]urea
N-{2-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}-4-(trifluoromethyl)benzamide
2-(4-fluorophenoxymethyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
(1S,4S)-5-(2-hydroxyacetyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
ethyl 3-benzyl-1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidine-3-carboxylate
2-methoxy-N-[(2R,3R)-2-methoxy-1'-propanoyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-2-amine
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-indole-2-carboxamide
N-methyl-6-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,6-dihydropyridine-3-carboxamide
ethyl 1-ethyl-5-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{5-[(3-phenylpiperidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}azocane
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2,4-dimethylpyrimidine
1-[(3-chlorophenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
3-{5-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridazine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(2-fluoro-4-methylphenyl)-3-[1-(thian-4-yl)piperidin-4-yl]urea
2-tert-butyl-N-(6-methoxyquinolin-8-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-[(3S,4R)-1-[3-(1H-imidazol-2-yl)benzoyl]-4-propylpyrrolidin-3-yl]acetamide
1-[2-methoxy-4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
2-oxo-N-phenyl-2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}acetamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-[(4-chlorophenyl)(phenyl)methyl]-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-(3-{[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}propyl)piperazin-2-one
4-hydroxy-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
4-(4-chlorophenyl)-1-[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]butan-1-one
6-[(2-fluorophenyl)methoxy]-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N,N-dimethyl-4-[3-(1H-pyrazol-3-yl)phenyl]-6-(trifluoromethyl)pyrimidin-2-amine
3-[(2-chlorophenyl)methyl]-N-[1-(thiophen-2-yl)propyl]-1,2-oxazole-5-carboxamide
(butan-2-yl)[(5-tert-butyl-1H-pyrazol-3-yl)methyl](pyridin-4-ylmethyl)amine