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1-ethyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methyl-1H-pyrazole-4-carboxamide
2-[4-(1,3-benzoxazol-2-yl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-hydroxyethyl)-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-methoxy-1-(3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidin-1-yl)ethan-1-one
1-[3-(3-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
ethyl 4-{[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]amino}piperidine-1-carboxylate
1-(2-methylphenyl)-4-(thiophene-3-carbonyl)-1,4-diazepane
N-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
(1S,5R)-3-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
4-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)carbamoyl]amino}-N-(2-methoxyethyl)benzamide
(1R,5S,6S)-6-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(furan-2-carbonyl)-N-(1-propyl-1H-1,2,4-triazol-3-yl)-1,4-diazepane-1-carboxamide
2-cyclopentanecarbonyl-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
9-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1,4-oxazepane-4-carboxamide
methyl 2-{1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-3-yl]-N-methylformamido}acetate
[2-(7-methyl-1H-indol-3-yl)ethyl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
4-[(3-cyclohexylpyrrolidin-1-yl)methyl]-1,3-thiazole
methyl 1-[(3R,5S)-5-(azepane-1-carbonyl)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(dimethylamino)methyl]-4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}phenol
2-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidine-3-carbonyl}pyridine
N-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
1-ethyl-8-[(4-hydroxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(diethylamino)ethyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4S)-1-[4-(5-methylfuran-2-yl)benzoyl]-4-propylpyrrolidin-3-amine
(2R)-2-[(6-methoxypyrimidin-4-yl)amino]-2-phenylethan-1-ol
4-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
3-{[2-(difluoromethoxy)phenyl]methyl}-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-(3-phenylpropyl)piperidin-3-yl}methanol
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-3-(pyridin-2-yl)propanamide
2-benzyl-N,1-dimethyl-5-propanamido-N-[1-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
4-(1H-imidazol-1-yl)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-4-carboxylic acid
N-(1,2-oxazol-3-ylmethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-methyl-5-[(1-propyl-1H-imidazol-2-yl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-methyl-2-[4-(piperidin-3-ylmethyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
4-(4-ethoxy-3-methylphenyl)-N-[2-(methylsulfamoyl)ethyl]-4-oxobutanamide
3-({1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}carbamoyl)pyridin-1-ium-1-olate
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
5-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
[(3-{[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-{1-ethyl-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
3-(2-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
N-methyl-N-[2-(2-methylphenyl)-1-[1-(naphthalene-2-carbonyl)piperidin-4-yl]ethyl]-2-(1H-pyrazol-1-yl)acetamide