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(1R,3S)-3-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)cyclopentane-1-carboxylic acid
6-butyl-2-(4-{[methyl(oxolan-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
7-fluoro-N-(propan-2-yl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
N-butyl-2-methyl-3-(1H-pyrazol-1-yl)-N-(thiophen-3-ylmethyl)propanamide
6-methyl-1-{3-oxo-3-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
4-{[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-(morpholin-4-yl)ethan-1-one
4-(2,3-difluoro-4-methoxybenzoyl)-2-ethyl-1-(propan-2-yl)piperazine
4-(5-chloro-2-methoxybenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
2-oxo-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-propylacetamide
5-[1-(2,1-benzoxazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[2-(dimethylamino)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-{1-[6-(4-hydroxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-2-oxo-N-phenylacetamide
5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
2-(2-{[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl]amino}ethyl)-6-phenyl-2,3-dihydropyridazin-3-one
3-[2-(methylsulfanyl)ethyl]-5-(oxolan-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
1-[4-({4-[ethyl(2-methylprop-2-en-1-yl)amino]quinazolin-2-yl}methyl)piperazin-1-yl]ethan-1-one
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
2-(cyclopentylmethyl)-N-(2-methoxyethyl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrimidine
1-[2-({[(2,5-difluorophenyl)methyl]amino}methyl)-4-methoxyphenoxy]-3-(dimethylamino)propan-2-ol
2-(pyrrolidin-1-yl)-4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinazoline
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-methyl-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1-propyl-1H-pyrazole
N,N-diethyl-1-(2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperidine-4-carboxamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amine
4-[5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-amino-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
1-(cyclopropylmethyl)-5-[2-(2-methoxyphenoxy)acetyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
2-hydroxy-2-(4-methoxyphenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]ethan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
2-(2,4-dimethoxyphenyl)-8-methoxy-5-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-{[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}-4-methyl-5,6,7,8-tetrahydroquinazoline
4-(4-chlorophenyl)-1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-ol
N-[(3S)-1-benzylpyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
ethyl 1-(cyclopent-1-ene-1-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-methoxy-1-{4-[2-(thiophen-2-yl)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carboxamide
4-fluoro-2-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)phenol
3-(4-methylpiperazin-1-yl)-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridazine
2-{4-[6-ethyl-4-(3-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
2-(azepan-1-yl)-2-(2,6-dimethoxypyridin-3-yl)acetic acid
1-(2-methoxy-5-{[(naphthalen-1-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol