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(2R)-2-hydroxy-3-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
N-(2-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
(2S,4S)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-(9H-fluoren-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroisoquinolin-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-oxo-N-(propan-2-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine
2-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
2-(cyclopropylmethyl)-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
8-[2-(2-chlorophenyl)-2-hydroxyacetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-cycloheptyl-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
methyl 2-{2-[(cyclopropylformamido)methyl]-5-methyl-2,3-dihydro-1-benzofuran-7-yl}benzoate
6-[({2-[(4-chlorophenyl)methoxy]ethyl}amino)methyl]-1,4-oxazepan-6-ol
2-cyclopropyl-4-phenyl-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{3-[3-(3-chloropyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
5-{5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
3-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}quinolin-7-ol
1-(4-methoxyphenyl)-3-methyl-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazole
ethyl 4-{4-[4-(tert-butylamino)piperidin-1-yl]benzoyl}piperazine-1-carboxylate
2-{[5-(4-acetylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-N-(propan-2-yl)acetamide
5-(azetidine-1-carbonyl)-3-(4-methoxyphenyl)-1H-pyrazole
N-[(2-chlorophenyl)methyl]-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
methyl 6-[3-(methylcarbamoyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]pyridine-2-carboxylate
4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-N-methyl-1,3-thiazol-2-amine
(3aR,6aS)-5-[(2-butyl-1H-imidazol-4-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1-hydroxypropan-2-yl)-1H-pyrazole-4-carboxamide
9-[2-(benzyloxy)ethyl]-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide
N-{[8-(quinolin-6-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]piperidine
1-[3-(2-phenylethyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)pyridine-3-carboxylic acid
(2S,4R)-1-[2-(furan-2-yl)-2-oxoacetyl]-N-methyl-4-(3-methylbutanamido)pyrrolidine-2-carboxamide
1-(4-cyano-2-ethylphenyl)-3-[1-(2,4-dimethoxyphenyl)ethyl]-3-methylurea
4-[2-(adamantan-1-yl)acetyl]-1-methylpiperazin-2-one
3-benzyl-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-chloro-4-fluorophenyl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N-(1-{4-[2,5-dioxo-4-(3-phenylpropyl)imidazolidin-4-yl]piperidin-1-yl}-3-methyl-1-oxobutan-2-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(cyclohexylsulfamoyl)-5-(1H-pyrazol-3-yl)benzamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-[3-(1-methyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-1-yl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-hydroxy-N,1-dimethylpiperidine-4-carboxamide
1-[2-(5-acetylthiophen-3-yl)acetyl]-4-methyl-1,4-diazepan-5-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-4-methyl-1,3-thiazole-5-carboxamide
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-benzyl-1-(2-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}thiophene-3-carboxamide
(1R,5S,8S)-8-methoxy-N-(2-phenylphenyl)-3-azabicyclo[3.2.1]octane-3-carboxamide
(1R,7S)-6-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one