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5-{2-[(2-methoxyethyl)amino]ethyl}-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]thiophene-3-carboxamide
7-[2-(2-fluorophenoxy)ethanesulfonyl]-2-oxa-7-azaspiro[4.5]decane
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-one
4-butyl-11-{[(4-phenyloxan-4-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-4-(4-{1-[2-(oxolan-3-yl)ethyl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
N5-[2-(3-chlorophenyl)ethyl]-N3-cyclohexyl-1-(2-methoxyethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{2-[2-(2-methoxyethyl)morpholin-4-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
(1R,5S,8R)-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2R)-oxolane-2-carbonyl]piperidine-4-carboxylic acid
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{2-[(2-aminopyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-cyclopentylpropan-1-one
2,3-dimethyl-7-(9H-purin-6-yl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propanamide
1-{3-oxo-3-[3-(2-phenylethyl)piperidin-1-yl]propyl}pyrrolidin-2-one
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
7-methoxy-4-methyl-2-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]quinazoline
3-(4-methoxyphenyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-[2-(2,4-difluorophenyl)-1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-methyl-4-oxobutanamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]oxane-4-carboxamide
(1S,5R)-3-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(2-fluorophenyl)ethyl]propanamide
4-(2-ethylphenyl)-6-methylpyrimidin-2-amine
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(trimethyl-1H-pyrazol-1-yl)propanamide
5-({5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}methyl)-1H-1,2,4-triazole
{3-propyl-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methanol
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(methylamino)pyridine-4-carboxamide
2-(2-hydroxyethyl)-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(oxolan-2-ylmethyl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
N-butyl-3-cyano-N-(3-phenylprop-2-yn-1-yl)benzamide
5-(3-methyl-1H-pyrazol-5-yl)-1-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-phenyl-1H-imidazole
1-{[1-(2-chlorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-1-(3,5-dimethylphenyl)piperazin-2-one
(3S,4S)-4-cyclopropyl-1-[2-(4-phenylpiperidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-butyl-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylpiperidine-3-carboxamide
7-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
9-methoxy-7-(2-methoxyphenyl)-4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(5-chloro-2,3-dimethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N,N,4-trimethyl-5-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}pyrimidin-2-amine
5-chloro-2-fluoro-N-methyl-N-[1-(pyridin-3-yl)ethyl]benzamide
N-benzyl-N-(cyclopropylmethyl)-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
3-ethyl-N,4-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]oxy}benzamide