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1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
5-(2,6-difluorophenoxymethyl)-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1,2-oxazole-3-carboxamide
2-(2-chlorophenyl)-3-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{4-[3-(5-methylfuran-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
2-phenyl-5-[4-(trifluoromethyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[(3R,4S)-4-(morpholin-4-yl)-1-(quinolin-6-ylmethyl)piperidin-3-yl]propanoic acid
12-[3-(morpholin-4-yl)piperidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
N,2-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-benzofuran-5-carboxamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]acetamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-[1-(1H-imidazol-1-yl)ethyl]-1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
1-(4-hydroxypiperidin-1-yl)-2-[4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]ethan-1-one
1-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
3-hydroxy-3-({[2-(1-hydroxycyclopentyl)ethyl]amino}methyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
4-(furan-2-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]benzamide
(2R,6R)-4-[3-(1H-imidazol-1-yl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-5-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-N-(2-phenylethyl)piperidin-4-amine
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
4-methanesulfonyl-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(piperidin-1-yl)-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
3-phenyl-8-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,8-diazaspiro[4.5]decan-2-one
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
1-(1-benzoylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyrrolidine-1-sulfonamide
3-[5-(2-hydroxybutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(2-methylbutyl)piperidin-4-ol
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
4-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
2-[3-(3,4-difluorophenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
methyl 3-(2-methoxybenzamido)-5-[(2-phenoxyacetamido)methyl]benzoate
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-hydroxypropyl)propanamide
{[(1R,5S,6R)-3-cyclopentanecarbonyl-3-azabicyclo[3.1.0]hexan-6-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
3-(4-chlorobenzoyl)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidine
N-{1-[2-(ethoxymethyl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl}acetamide
[2-fluoro-5-(5-methyl-1,3-benzoxazol-2-yl)phenyl]methanol
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(quinoxalin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-butyl-4-({3-[1-(dimethylamino)ethyl]phenyl}methyl)piperazin-2-one
ethyl 1-methanesulfonyl-4-(2-phenoxyethyl)piperidine-4-carboxylate
4-[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-imidazol-2-yl]-N-methylbenzene-1-sulfonamide
2-chloro-4-[4-(1-hydroxypropyl)phenyl]benzamide
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-[(3-chlorophenyl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5,6-dimethyl-2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-ethyl-8-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one