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4-phenoxy-1-[3-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
2-(2,3-difluorophenyl)-N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}acetamide
4-(1-butyl-1H-imidazol-2-yl)-3,5-dimethylphenol
N-benzyl-6-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-(4-fluorophenyl)-1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]butan-1-one
4-(2,3-dihydro-1H-isoindol-2-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]butanamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
4-[(2S,4R)-1-[(3,4-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
N,3,5-trimethyl-N-(2-methylprop-2-en-1-yl)adamantane-1-carboxamide
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
(2S,4R)-4-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamido]-N,N-diethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-methyl-5-{4-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-3-(1H-pyrazol-4-yl)benzamide
N-[2-(2-chlorophenyl)ethyl]-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
N-[(1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[2-(3,4-dimethoxyphenyl)ethyl]methylamine
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-amino-N-butyl-4-methyl-N-[(2-methylphenyl)methyl]pyrimidine-5-carboxamide
N-(1-{1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
7-(1,3-benzothiazol-2-yl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(2,4-difluorophenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydro-1H-inden-2-amine
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
2-methyl-N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
4,5-dimethyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-2-(1H-1,2,3,4-tetrazol-1-yl)thiophene-3-carboxamide
N-{[8-(2,6-dimethylhept-5-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
3-(3-methoxypropyl)-1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]piperidine-3-carboxylic acid
(1S,5R)-3-cyclobutanecarbonyl-N-(3,4-difluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(4-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
3-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyridazine
3-(2H-1,3-benzodioxol-5-yl)-1-{[2-(diethylamino)pyridin-3-yl]methyl}urea
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
(2S)-N-[3-(3-chlorophenyl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
ethyl 2-(1-{1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
4'-(3-phenoxypropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(4-fluorophenyl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-(piperidin-1-yl)ethan-1-one
N-tert-butyl-2-(6-cyclopropylpyrimidin-4-yl)benzene-1-sulfonamide
5-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-1H-1,3-benzodiazole
4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
ethyl 5-({[7-oxo-2-(2-phenylacetamido)-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl]formamido}methyl)furan-2-carboxylate
2-(cyclopentylmethyl)-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
4-(furan-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(5-methylpyridin-3-yl)benzamide
(2S)-2-amino-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-cyclohexylethan-1-one
3-chloro-N-(2-methoxyethyl)-4-({1-[1-(propan-2-yl)piperidin-4-yl]piperidin-4-yl}oxy)benzamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide