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(3R,9aR)-3-benzyl-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-3-[3-(methylsulfanyl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[7-(cyclohex-3-en-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}pyridine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(4-fluoro-3-methylphenyl)urea
N-cyclopropyl-3-[1-(6-ethyl-2-methylquinoline-4-carbonyl)piperidin-4-yl]propanamide
1-cycloheptanecarbonyl-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(pyridin-3-yloxy)propyl]propanamide
1-{6-[(4-fluorophenyl)methoxy]-3-oxo-4-(propan-2-yl)-1,4-diazepan-1-yl}-2-phenylethane-1,2-dione
(5-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-indole-6-carboxamide
N-{2-[4-({[(4-methoxy-2,5-dimethylphenyl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-methoxy-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
N-methyl-3-(piperidin-4-ylmethyl)-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
(3aS,6aR)-5-{[3-(methylsulfanyl)phenyl]methyl}-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-methyl-N-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}cyclohexanamine
ethyl 3-[(4-fluorophenyl)methyl]-1-[2-(furan-2-yl)-2-oxoacetyl]piperidine-3-carboxylate
N-(2,3-dimethylphenyl)-2-[(2-methoxyethyl)(1-methylpiperidin-4-yl)amino]acetamide
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-(3-hydroxy-3-phenylpropyl)-1-methylurea
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-[2-(1H-indol-3-yl)ethyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-{3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}propanamide
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(2-phenoxypropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
2-(dimethylamino)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(4-fluorophenyl)acetamide
2-{4-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
(4aS,8aR)-6-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
14-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-amino-4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(2-methoxyethyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(2-methyl-1,3-benzothiazol-6-yl)urea
(3aR,6aR)-2-acetyl-5-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(2-ethoxyethyl)pyrimidin-2-amine
N'-(2-ethylphenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]ethanediamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine-4-carboxamide
8-[(5-acetylthiophen-3-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(1H-imidazol-1-yl)propyl]-2-(2-oxopiperidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
1-[1'-(5-propyl-1,3,4-thiadiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-(4-benzoylpiperidin-1-yl)-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(1H-indol-1-yl)ethyl]propanamide
3-cyclopropyl-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
2-(methylsulfanyl)-4-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine-5-carboxylic acid
4-(3-ethyl-1,2-oxazole-5-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
5-ethanesulfonamido-N-(1H-imidazol-2-ylmethyl)-N,1-dimethyl-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-(pentan-3-yl)piperazin-2-yl}ethan-1-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
2-methoxy-4-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1,3-thiazole-5-carboxamide
(3S,4R)-1-(4-fluoro-2-methylbenzenesulfonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol